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Patent Searching and Data


Title:
不安及び痙攣の治療のための7-TERT-ブチル-3-(2-フルオロフェニル)-6-(2H-(1,2,4)トリアゾール-3-イルメトキシ)-(1,2,4)トリアゾロ(4,3-B)ピリダジン
Document Type and Number:
Japanese Patent JP2005507391
Kind Code:
A
Abstract:
The compound (I) is a GABAa receptor ligand, functionally selective for the alpha2 and/or alpha3 subunit, and is useful in the treatment of deleterious mental states, in particular anxiety.

Inventors:
Carling, William Robert
Moore, Kevin William
Street, Leslie Yogyov
Application Number:
JP2003528815A
Publication Date:
March 17, 2005
Filing Date:
September 13, 2002
Export Citation:
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Assignee:
Merck Sharp End Dome Limited
International Classes:
A61K31/519; A61P25/00; A61P25/08; A61P25/22; C07D487/04; (IPC1-7): C07D487/04; A61K31/519; A61P25/08; A61P25/22
Attorney, Agent or Firm:
Yoshio Kawaguchi
Akio Ichiiri
Makoto Ono
Katsuma Osaki
Mitsuaki Tsubokura