Title:
ブラジキニンB1アンタゴニストとしての新規なキノキサリノン誘導体
Document Type and Number:
Japanese Patent JP2006511550
Kind Code:
A
Abstract:
2-Quinoxalinone derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
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Inventors:
Sue, Dice
Bock, Mark Gee
Bock, Mark Gee
Application Number:
JP2004560735A
Publication Date:
April 06, 2006
Filing Date:
December 09, 2003
Export Citation:
Assignee:
MERCK & COMPANY INCOPORATED
International Classes:
C07D403/06; A61K31/498; A61K31/5377; A61P1/04; A61P1/18; A61P11/00; A61P11/06; A61P13/10; A61P17/02; A61P19/02; A61P19/06; A61P19/08; A61P25/04; A61P27/02; A61P27/16; A61P29/00; A61P35/00; A61P43/00; C07D401/12; C07D403/12; C07D405/12; C07D409/14; C07D471/04
Attorney, Agent or Firm:
Yoshio Kawaguchi
Makoto Ono
Katsuma Osaki
Mitsuaki Tsubokura
Makoto Ono
Katsuma Osaki
Mitsuaki Tsubokura