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Title:
電位型イオンチャネルの調節因子としての二環式誘導体
Document Type and Number:
Japanese Patent JP2009507851
Kind Code:
A
Abstract:
Bicyclic derivatives useful as ion channel antagonists are disclosed herein. The compositions thereof are useful for treating or relieving pain-related conditions.

Inventors:
Neubert, Timothy
Zimmerman, Nicole
Kawatokar, Altis
Martinborough, Esther
Termin, Andreas
Application Number:
JP2008530198A
Publication Date:
February 26, 2009
Filing Date:
September 08, 2006
Export Citation:
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Assignee:
VERTEX PHARMACEUTICALS INCORPORATED
International Classes:
C07D277/20; A61K31/426; A61K31/427; A61K31/4709; A61P1/00; A61P5/00; A61P9/06; A61P13/02; A61P19/02; A61P21/00; A61P25/00; A61P25/04; A61P25/06; A61P25/08; A61P25/14; A61P25/22; A61P25/24; A61P25/28; A61P29/00; A61P29/02; A61P43/00; C07D277/52; C07D417/12
Domestic Patent References:
JP2007501804A2007-02-01
JP2003055209A2003-02-26
JP2005526137A2005-09-02
Foreign References:
WO2000071506A22000-11-30
US5378715A1995-01-03
US20050085518A12005-04-21
Other References:
JPN6012022920; J. Med. Chem. vol.40, no.6, 1997, p.996-1004
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita