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Title:
ピラゾロン誘導体のエマルジョン製剤
Document Type and Number:
Japanese Patent JP2011504177
Kind Code:
A
Abstract:
Pyrazolone derivative emulsion formulations are provided. The emulsion formulations include a pyrazolone derivative active agent, e.g., Edaravone, oil, water and an emulsifier. Also provided are methods of making and using the subject emulsion formulations.

Inventors:
Kiichiro Nabeta
Application Number:
JP2010535000A
Publication Date:
February 03, 2011
Filing Date:
November 07, 2008
Export Citation:
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Assignee:
Teikoku Pharma USA Inc.
Techno Guard Co., Ltd.
International Classes:
A61K31/4152; A61K9/107; A61K47/24; A61K47/44; A61P7/10; A61P9/10; A61P21/00; A61P21/02; A61P35/00; C07D231/26
Domestic Patent References:
JPS52145525A1977-12-03
JP2006052172A2006-02-23
JPS52145525A1977-12-03
JP2006052172A2006-02-23
Foreign References:
WO2002000260A12002-01-03
CN1440749A2003-09-10
WO2002092082A12002-11-21
WO2002000260A12002-01-03
CN1440749A2003-09-10
WO2002092082A12002-11-21
Other References:
JPN6013017487; 新・ドラッグデリバリーシステム pp.136-143, 20000131, 株式会社シーエムシー  島  健太郎
JPN6013017487; 新・ドラッグデリバリーシステム pp.136-143, 20000131, 株式会社シーエムシー  島  健太郎
CSNC200900984014; 新・ドラッグデリバリーシステム pp.136-143, 20000131, 株式会社シーエムシー  島  健太郎
Attorney, Agent or Firm:
Kyousei Tamura
Samejima Mutsumi
Masahiro Nitta
Yushiro Tsuboi