Title:
新規TRPV3モジュレーター
Document Type and Number:
Japanese Patent JP2013538800
Kind Code:
A
Abstract:
Disclosed herein are modulators of TRPV3 of formula (I) wherein G1, X1, X2, X3, X4, X5, G2, Z1, Ra, Rb, u, and p are as defined in the specification. Compositions comprising such compounds and methods for treating conditions and disorders using such compounds and compositions are also presented.
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Inventors:
Bybert eror kay
Clapham, Bruce
Cocks, Filly Bee
Danen, Jerome F
Gomutsuyan, Arthur
Court, michael yee
Kim, Philip Earl
Voight, Eric A.
Clapham, Bruce
Cocks, Filly Bee
Danen, Jerome F
Gomutsuyan, Arthur
Court, michael yee
Kim, Philip Earl
Voight, Eric A.
Application Number:
JP2013523450A
Publication Date:
October 17, 2013
Filing Date:
August 10, 2010
Export Citation:
Assignee:
AbbVie Incorporated
International Classes:
C07D213/30; A61K31/4402; A61K31/4433; A61K31/505; A61K31/5377; A61P25/04; C07D213/42; C07D239/26; C07D401/12; C07D405/06
Domestic Patent References:
JP2013532177A | 2013-08-15 | |||
JPH02295972A | 1990-12-06 | |||
JP2002502844A | 2002-01-29 | |||
JP2005528385A | 2005-09-22 | |||
JPS6471830A | 1989-03-16 | |||
JPH09500875A | 1997-01-28 | |||
JP2006508130A | 2006-03-09 | |||
JP2009520808A | 2009-05-28 | |||
JPH04235966A | 1992-08-25 | |||
JPS60109539A | 1985-06-15 | |||
JPH08511010A | 1996-11-19 | |||
JPS60230742A | 1985-11-16 | |||
JPS54138547A | 1979-10-27 |
Foreign References:
WO2010110231A1 | 2010-09-30 | |||
CN1215715A | 1999-05-05 | |||
WO2009115427A1 | 2009-09-24 |
Other References:
JPN6014040540; TETRAHEDRON LETTERS Vol.28, No.50, 1987, pp.6313-6316
JPN6014040542; TETRAHEDRON Vol.59, 2003, pp.8525-8542
JPN6014040544; J.ORG.CHEM. Vol.66, 2001, pp.4450-4452
JPN6014040548; JOURNAL OF MEDICINAL CHEMISTRY Vol.10, No.1, 1967, pp.128-129
JPN6014040549; JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol.79, 1957, pp.472-480
JPN6014040551; JOURNAL OF MEDICINAL CHEMISTRY Vol.17, No.11, 1974, pp.1188-1193
JPN6014040553; HUANAN NONGYE DAXUE XUEBAO (JOURNAL OF SOUTH CHINA AGRICULTURAL UNIVERSITY) Vol.26, No.1, 2005, pp.67-69
JPN6014040554; JOURNAL OF ORGANIC CHEMISTRY Vol.18, 1953, pp.1058-1064
JPN6014040555; JOURNAL OF HETEROCYCLIC CHEMISTRY Vol.18, No.4, 1981, pp.815-820
JPN6014040558; JOURNAL OF MEDICINAL CHEMISTRY Vol.30, No.6, 1987, pp.1054-1068
JPN6014040559; EGYPTIAN JOURNAL OF CHEMISTRY Vol.18, No.3, 1975, pp.581-586
JPN6014040560; JOURNAL OF ORGANIC CHEMISTRY Vol.37, No.2, 1972, pp.173-178
JPN6014040542; TETRAHEDRON Vol.59, 2003, pp.8525-8542
JPN6014040544; J.ORG.CHEM. Vol.66, 2001, pp.4450-4452
JPN6014040548; JOURNAL OF MEDICINAL CHEMISTRY Vol.10, No.1, 1967, pp.128-129
JPN6014040549; JOURNAL OF THE AMERICAN CHEMICAL SOCIETY Vol.79, 1957, pp.472-480
JPN6014040551; JOURNAL OF MEDICINAL CHEMISTRY Vol.17, No.11, 1974, pp.1188-1193
JPN6014040553; HUANAN NONGYE DAXUE XUEBAO (JOURNAL OF SOUTH CHINA AGRICULTURAL UNIVERSITY) Vol.26, No.1, 2005, pp.67-69
JPN6014040554; JOURNAL OF ORGANIC CHEMISTRY Vol.18, 1953, pp.1058-1064
JPN6014040555; JOURNAL OF HETEROCYCLIC CHEMISTRY Vol.18, No.4, 1981, pp.815-820
JPN6014040558; JOURNAL OF MEDICINAL CHEMISTRY Vol.30, No.6, 1987, pp.1054-1068
JPN6014040559; EGYPTIAN JOURNAL OF CHEMISTRY Vol.18, No.3, 1975, pp.581-586
JPN6014040560; JOURNAL OF ORGANIC CHEMISTRY Vol.37, No.2, 1972, pp.173-178
Attorney, Agent or Firm:
Kawaguchi International Patent Office