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Title:
選択的FAK阻害剤
Document Type and Number:
Japanese Patent JP2014505719
Kind Code:
A
Abstract:
A compound of the formula (I): where R1 or R2 is a cyclc amine group and R5 is an aromatic group with a carbonyl containing substituent for use as a FAK inhibitor.

Inventors:
Ian Peter Holmes
Irva Bergman
Gillian Elizabeth Lunis
Marika Nikak
Neil Choi
Catherine Faye Hemley
Scott Raymond Walker
Richard Charles Voithick
Danny Ganeim
Romina Ressen
Application Number:
JP2013553996A
Publication Date:
March 06, 2014
Filing Date:
February 17, 2012
Export Citation:
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Assignee:
CANCER THERAPEUTICS CRC PTY LIMITED
International Classes:
C07D239/42; A61K31/505; A61K31/506; A61P35/00; A61P43/00; C07D401/12
Domestic Patent References:
JP2013534227A2013-09-02
JP2006515298A2006-05-25
JP2005509624A2005-04-14
JP2006520354A2006-09-07
JP2013534227A2013-09-02
JP2006515298A2006-05-25
JP2005509624A2005-04-14
JP2006520354A2006-09-07
Foreign References:
WO2010058030A12010-05-27
WO2010055117A12010-05-20
WO2010058030A12010-05-27
WO2010055117A12010-05-20
Attorney, Agent or Firm:
Axis International Patent Business Corporation



 
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