Title:
カテコールO−メチルトランスフェラーゼ活性阻害化合物
Document Type and Number:
Japanese Patent JP2015522547
Kind Code:
A
Abstract:
式(I)(式中、R1は、特許請求の範囲において定義したものである)の化合物は、COMT酵素阻害活性を示し、したがって、COMT阻害剤として有用である。
Inventors:
Aalmark, Marco
Dimbell, David
Kauppara, Mika
Ruilo, Anne
Payunen, Taina
Pustunen, Yarmo
Chiainen, Aiya
Vicemers, matches
Messinger, Joseph
Dimbell, David
Kauppara, Mika
Ruilo, Anne
Payunen, Taina
Pustunen, Yarmo
Chiainen, Aiya
Vicemers, matches
Messinger, Joseph
Application Number:
JP2015513234A
Publication Date:
August 06, 2015
Filing Date:
May 23, 2013
Export Citation:
Assignee:
Orion Corporation
International Classes:
C07C255/53; A61K31/198; A61K31/275; A61K31/341; A61K31/343; A61K31/351; A61K31/381; A61K31/40; A61K31/402; A61K31/415; A61K31/428; A61K31/4406; A61K31/4409; A61K31/451; A61K31/5375; A61K31/5377; A61K45/00; A61P25/16; A61P43/00; C07C255/54; C07C255/57; C07C255/59; C07C311/29; C07C317/22; C07C317/46; C07C323/62; C07D207/337; C07D211/14; C07D213/57; C07D213/70; C07D231/12; C07D265/30; C07D277/74; C07D295/14; C07D295/18; C07D307/54; C07D307/78; C07D307/79; C07D309/20; C07D333/24; C07D333/28; C07D333/32; C07D333/36; C07D333/60
Domestic Patent References:
JPS62240649A | 1987-10-21 | |||
JPH11505821A | 1999-05-25 | |||
JP2012051884A | 2012-03-15 | |||
JP2009508968A | 2009-03-05 |
Foreign References:
WO2007063789A1 | 2007-06-07 |
Attorney, Agent or Firm:
Asahina Patent Office