Title:
フルオロケトライドを調製するための方法
Document Type and Number:
Japanese Patent JP2018508537
Kind Code:
A
Abstract:
フルオロケトライド化合物を調製するための方法及び中間体を本明細書で記載する。【選択図】なし
Inventors:
David Eugene, Pereira
Schneider, Stephanie.
Deo, Keshav
Schneider, Stephanie.
Deo, Keshav
Application Number:
JP2017546856A
Publication Date:
March 29, 2018
Filing Date:
March 05, 2016
Export Citation:
Assignee:
Sempura Pharmaceuticals, Inc.
International Classes:
C07H17/08; A61K31/7056; A61P31/04; A61P33/02
Domestic Patent References:
| JP2011500834A | 2011-01-06 | |||
| JP2014507447A | 2014-03-27 |
Foreign References:
| US20060100164A1 | 2006-05-11 | |||
| US20080096828A1 | 2008-04-24 |
Other References:
DENIS, A. ET AL.: "B-keto-ester chemistry and ketolides. Synthesis and antibacterial activity of 2-halogeno, 2-methyl a", BIOORG. MED. CHEM. LETT., vol. 10, JPN6020000044, 2000, pages 2019 - 2022, XP004214160, ISSN: 0004189780, DOI: 10.1016/S0960-894X(00)00392-9
KANEKO, T. ET AL.: "Novel tethers in ketolide antibiotics", BIOORG. MED. CHEM. LETT., vol. Vo.17, JPN6020000045, 2007, pages 5049 - 5053, ISSN: 0004189781
XU, X. ET AL.: "Synthesis and antibacterial activity of C2-fluoro, C6-carbamate ketolides, and their C9-oximes", BIOORG. MED. CHEM. LETT., vol. Vo.15, JPN6020000046, 2005, pages 883 - 887, ISSN: 0004189782
ZHU, J. Z. ET AL.: "Structure-activity relationships of macrolides against mycobacterium tuberculosis", TUBERCULOSIS, vol. 88, JPN6020000047, 2008, pages 49 - 63, ISSN: 0004189783
KANEKO, T. ET AL.: "Novel tethers in ketolide antibiotics", BIOORG. MED. CHEM. LETT., vol. Vo.17, JPN6020000045, 2007, pages 5049 - 5053, ISSN: 0004189781
XU, X. ET AL.: "Synthesis and antibacterial activity of C2-fluoro, C6-carbamate ketolides, and their C9-oximes", BIOORG. MED. CHEM. LETT., vol. Vo.15, JPN6020000046, 2005, pages 883 - 887, ISSN: 0004189782
ZHU, J. Z. ET AL.: "Structure-activity relationships of macrolides against mycobacterium tuberculosis", TUBERCULOSIS, vol. 88, JPN6020000047, 2008, pages 49 - 63, ISSN: 0004189783
Attorney, Agent or Firm:
Ryoichi Takaoka
Nao Oda
Akiyo Iwahori
Kaoru Takahashi
Nao Oda
Akiyo Iwahori
Kaoru Takahashi