Title:
新規なフェロポーチン阻害剤
Document Type and Number:
Japanese Patent JP2018536641
Kind Code:
A
Abstract:
本発明は、一般式(I)の新規なフェロポーチン阻害剤、それらを含む医薬組成物、並びに特にヘプシジン欠如又は鉄代謝障害によって引き起こされる疾患、例えば特に鉄過剰状態、例えば特にサラセミア及びヘモクロマトーシスを予防及び/又は治療するための医薬品としてのその使用に関する。【選択図】図1
Inventors:
Durenberger, Franz
Boer, Wirm
Burghard, Susanna
Burgert, michael
Alice, Calogerakis
Lime, stephan
Manorova, Vania
Voice, susan
Yarnold, Christopher John
Pena, Paula
John the Shepherd
Lexi, Christina
Jar Jess-Pike, Richard
John Scott
Boer, Wirm
Burghard, Susanna
Burgert, michael
Alice, Calogerakis
Lime, stephan
Manorova, Vania
Voice, susan
Yarnold, Christopher John
Pena, Paula
John the Shepherd
Lexi, Christina
Jar Jess-Pike, Richard
John Scott
Application Number:
JP2018520090A
Publication Date:
December 13, 2018
Filing Date:
October 21, 2016
Export Citation:
Assignee:
Vifor (International) AG
International Classes:
C07D235/14; A61K31/4184; A61K31/426; A61K31/427; A61K31/437; A61K31/4375; A61K31/4439; A61K31/444; A61K31/4725; A61K31/501; A61K31/5025; A61K31/506; A61K31/5377; A61K45/00; A61K45/06; A61P1/16; A61P3/00; A61P7/00; A61P7/06; A61P9/00; A61P25/16; A61P25/28; A61P29/00; A61P31/04; A61P43/00; C07D277/56; C07D401/14; C07D413/14; C07D417/12; C07D417/14; C07D471/04; C07D487/04; C07D495/04
Domestic Patent References:
JP2005514330A | 2005-05-19 | |||
JP2008542276A | 2008-11-27 | |||
JP2010513493A | 2010-04-30 | |||
JP2018535203A | 2018-11-29 |
Foreign References:
WO2011029832A1 | 2011-03-17 |
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yousuke Kawasaki
Takuya Gomibuchi
Toshikazu Imato
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Yoshikazu Iwase
Yasufumi Shiroyama
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yousuke Kawasaki
Takuya Gomibuchi
Toshikazu Imato
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Yoshikazu Iwase
Yasufumi Shiroyama