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Patent Searching and Data


Title:
CHEMICAL COMPOUND USEFUL AS INTERMEDIATE FOR PREPARING A CATECHOL-O-METHYLTRANSFERASE INHIBITOR
Document Type and Number:
Japanese Patent JP2020059729
Kind Code:
A
Abstract:
To provide a methylated intermediate which may be demethylated to provide an inhibitor of catechol-O-methyltransferase useful in the treatment of Parkinson's disease, and to provide methods of producing and using the intermediate.SOLUTION: There are provided a compound of formula (I), and methods of producing and using the intermediate.SELECTED DRAWING: None

Inventors:
DOMENICO RUSSO
LASZLO ERNO KISS
JORGE BRUNO REIS WAHNON
DAVID ALEXANDER LEARMONTH
TIBOR ESZENYI
AXEL ZIMMERMANN
BJOERN SCHLUMMER
MICHAEL KREIS
KLAUS REITER
Application Number:
JP2019214566A
Publication Date:
April 16, 2020
Filing Date:
November 27, 2019
Export Citation:
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Assignee:
NOVIPHARMA SA
International Classes:
C07D413/04; A61K9/14; A61K31/198; A61K31/4439; A61K45/00; A61P25/16; A61P43/00
Attorney, Agent or Firm:
Seiji Ohno
Yuko Matsuniya
Umeda Shinsuke