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Title:
【発明の名称】複数層の制御放出処方剤
Document Type and Number:
Japanese Patent JP3426230
Kind Code:
B2
Abstract:
Controlled release pharmaceutical beads are provided having a multi-layered core and a multi-layered periphery. The core contains at least (A) an inner portion having a suitable organic acid and (B) a sustainably-acid-releasing coating thereover. The periphery contains at least (A) an inner portion having a mixture of at least (i) a pharmaceutical compound and (ii) a surface-active agent, and (B) a sustainably-drug-releasing exterior coating.

Inventors:
Kazuo Noda
Kousuke Yoshino
Yoshiyuki Hirakawa
McLaren, David, Dee.
Skartetie, Paul, F.
Leffler, John, Earl.
Beck, Greg, M.
Application Number:
JP50028993A
Publication Date:
July 14, 2003
Filing Date:
May 20, 1992
Export Citation:
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Assignee:
Aventis Pharmaceuticals Incorporated
Tanabe Pharmaceutical Co., Ltd.
International Classes:
A61K9/50; A61K9/54; A61K9/58; A61K31/554; A61K47/12; A61K47/20; A61K9/52; A61P9/12; (IPC1-7): A61K9/52; A61K31/554; A61K47/12; A61K47/20; A61P9/12
Domestic Patent References:
JP56103111A
JP63227519A
JP5315411A
JP37238A
Attorney, Agent or Firm:
Katsuro Sasai