Title:
1, 2-imidazo [a] pyridine compound
Document Type and Number:
Japanese Patent JP6211556
Kind Code:
B2
Abstract:
Imidazo[1,2-a]pyridines are disclosed. Compounds of the invention are useful therapeutic agents and their inclusion in pharmaceutical formulations and use in methods of treatment are disclosed. Many of the compounds disclosed herein may be represented by the following generic formula: in which Y is a direct bond or heteroatom and A3 is usually a nitrogenous heterocycle.
Inventors:
Fan, kun kevin
U, Frank Shinhe
Glover, Paul Tee.
Hopkins, Cessie.
Campbell, Una
Sicily, Milan
Spear, Kelly El.
U, Frank Shinhe
Glover, Paul Tee.
Hopkins, Cessie.
Campbell, Una
Sicily, Milan
Spear, Kelly El.
Application Number:
JP2015090193A
Publication Date:
October 11, 2017
Filing Date:
April 27, 2015
Export Citation:
Assignee:
Sunovion Pharmaceuticals Inc.
International Classes:
C07D487/04; A61K31/5025; A61K31/513; A61K31/52; A61K31/522; A61P1/08; A61P25/04; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P27/02; A61P43/00; C07D519/00
Domestic Patent References:
| JP2004506633A | ||||
| JP2007509960A | ||||
| JP61047485A |
Foreign References:
| WO2006128692A1 | ||||
| WO2006128693A1 | ||||
| EP1845098A1 | ||||
| WO1989001333A1 | ||||
| WO2002002557A1 | ||||
| WO2007110438A1 | ||||
| WO2008022396A1 | ||||
| GB1135893B | ||||
| CA1263390C | ||||
| WO2008116665A1 | ||||
| WO2006101455A1 | ||||
| WO2005080355A1 |
Other References:
ZHAI, XIN ET AL,Synthesis and antibacterial activity of novel oxazolidinone analogs containing substituted thiazole/fused-bicyclic groups,Chemical Research in Chinese Universities,2006年,22(4),459-464
BARLIN, GORDON B. ET AL,Imidazo[1,2-b]pyridazines. X. Syntheses and central nervous system activities of some 3-(acetamido, benzamido, substituted benzamido or dimethylamino)methyl-2-(phenyl or substituted phenyl)-6-(halo, alkylthio, alkoxy, phenylthio, phenoxy, benzylthio or benzyloxy)imidazo[1,2-b]pyridazines,Australian Journal of Chemistry,1992年,45(4),731-49
ENGUEHARD CECILE,SYNTHESIS OF DIARYL-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINES DESIGNED AS POTENTIAL AROMATASE INHIBITORS,CHEMICAL & PHARMACEUTICAL BULLETIN,2000年,V48 N7,P935-940
C.G.WERMUTH編,『最新 創薬化学 上巻』,株式会社テクノミック,1998年 8月15日,235-271頁,13章 等価置換に基づく分子の変換
COLLINS, JON L. ET AL,N-(2-Benzoylphenyl)-L-tyrosine PPAR.gamma. Agonists. 2. Structure-Activity Relationship and Optimization of the Phenyl Alkyl Ether Moiety,JOURNAL OF MEDICINAL CHEMISTRY,1998年,41(25),5037-5054
BARLIN, GORDON B. ET AL,Imidazo[1,2-b]pyridazines. X. Syntheses and central nervous system activities of some 3-(acetamido, benzamido, substituted benzamido or dimethylamino)methyl-2-(phenyl or substituted phenyl)-6-(halo, alkylthio, alkoxy, phenylthio, phenoxy, benzylthio or benzyloxy)imidazo[1,2-b]pyridazines,Australian Journal of Chemistry,1992年,45(4),731-49
ENGUEHARD CECILE,SYNTHESIS OF DIARYL-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINES DESIGNED AS POTENTIAL AROMATASE INHIBITORS,CHEMICAL & PHARMACEUTICAL BULLETIN,2000年,V48 N7,P935-940
C.G.WERMUTH編,『最新 創薬化学 上巻』,株式会社テクノミック,1998年 8月15日,235-271頁,13章 等価置換に基づく分子の変換
COLLINS, JON L. ET AL,N-(2-Benzoylphenyl)-L-tyrosine PPAR.gamma. Agonists. 2. Structure-Activity Relationship and Optimization of the Phenyl Alkyl Ether Moiety,JOURNAL OF MEDICINAL CHEMISTRY,1998年,41(25),5037-5054
Attorney, Agent or Firm:
Kenichi Morita
Kenjiro Yamaguchi
Kenjiro Yamaguchi