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Title:
レニン阻害剤としての1-アシルアミノ-2-ヒドロキシ-3-アミノ-ω-アリールアルカン
Document Type and Number:
Japanese Patent JP2008528691
Kind Code:
A
Abstract:
1-Acylamino-2-hydroxy-3-amino-omega-arylalkanes of formula I. and the salts thereof, have renin-inhibiting properties and can be used as antihypertensive, medicinally active ingredients.

Inventors:
McGeehan, Gerrard
Simpson, Robert Dee.
Twen, Wenyuan
Baldwin, John Jay.
Claremon, David A.
Dillard, Lawrence W..
Ishchenko, Alexei Buoy.
Yuan, Chin
Shu, Chen Long
Kakatian, slavation
Tice, Colin
Chao, Way
Application Number:
JP2007554177A
Publication Date:
July 31, 2008
Filing Date:
February 01, 2006
Export Citation:
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Assignee:
Vite Pharmaceuticals, Inc.
International Classes:
C07C233/36; A61K31/164; A61K31/17; A61K31/18; A61K31/27; A61K31/336; A61K31/421; A61K31/4453; A61K45/00; A61P5/42; A61P9/00; A61P9/04; A61P9/12; A61P13/12; A61P25/22; A61P25/28; A61P27/02; A61P27/06; A61P35/00; A61P43/00; C07C233/62; C07C271/12; C07C275/24; C07C307/06; C07C311/13; C07C335/12; C07D263/06; C07D295/18; C07D301/06; C07D303/36
Foreign References:
US5627182A1997-05-06
WO2003050073A12003-06-19
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita