Title:
1,3-ジ置換された4-メチル-1H-ピロール-2-カルボン酸アミド及び医薬を製造するためのその使用
Document Type and Number:
Japanese Patent JP5156011
Kind Code:
B2
Abstract:
1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides corresponding to formula I methods for their production, pharmaceutical compositions containing them, and the use thereof for noradrenalin receptor regulation, particularly for inhibiting noradrenalin reuptake, and/or for 5-HT receptor regulation, particularly for inhibiting 5-hydroxy tryptophan reuptake, and/or for opioid receptor regulation and/or for batrachotoxin (BTX) receptor regulation and/or for treating or inhibiting pain and other conditions.
Inventors:
Oberberch Stefan
Zunderman Bernd
Zunderman Corinna
Bestelfeld Edwald
Hennies Hagen-Heinrich
Zunderman Bernd
Zunderman Corinna
Bestelfeld Edwald
Hennies Hagen-Heinrich
Application Number:
JP2009513607A
Publication Date:
March 06, 2013
Filing Date:
June 08, 2007
Export Citation:
Assignee:
Grunenthal Gesellschaft Mito Beschlenktel Haftung
International Classes:
C07D207/34; A61K31/40; A61K31/4025; A61K31/404; A61K31/4178; A61K31/4439; A61K31/454; A61K31/496; A61K31/5377; A61P1/12; A61P3/04; A61P7/10; A61P7/12; A61P9/00; A61P11/14; A61P13/10; A61P15/10; A61P17/04; A61P23/02; A61P25/00; A61P25/04; A61P25/06; A61P25/08; A61P25/14; A61P25/16; A61P25/22; A61P25/24; A61P25/26; A61P25/28; A61P25/32; A61P25/36; A61P43/00; C07D401/06; C07D401/12; C07D403/06; C07D403/12; C07D405/04; C07D409/12
Domestic Patent References:
| JP2003252854A | ||||
| JP2006501243A | ||||
| JP11322711A | ||||
| JP4502146A |
Foreign References:
| WO2004108685A1 | ||||
| WO2005113497A1 |
Attorney, Agent or Firm:
Mitsufumi Esaki
Blacksmith
Blacksmith