Login| Sign Up| Help| Contact|

Patent Searching and Data


Title:
3-アミノアルキル-1,4-ジアゼパン-2-オンメラノコルチン-5受容体アンタゴニスト
Document Type and Number:
Japanese Patent JP5503557
Kind Code:
B2
Abstract:
The present invention provides compounds of Formula (I) that are useful for modulating the biological activity of the melanocortin-5 receptor (MC5R). Compounds of this invention can be used to treat diseases and/or conditions in which downregulation of MC5R is beneficial. Such diseases and/or conditions include, but are not limited to, acne, seborrhea, seborrheic dermatitis, cancer, and inflammatory diseases.

Inventors:
Blaskovich, Mark, Arnold, Thomas
Cassidy, Peter, Joseph
Application Number:
JP2010547917A
Publication Date:
May 28, 2014
Filing Date:
February 27, 2009
Export Citation:
Click for automatic bibliography generation   Help
Assignee:
MIMETICA PTY LTD
International Classes:
C07D243/08; A61K31/551; A61P17/00; A61P43/00; C07D401/04; C07D401/06; C07D401/12; C07D403/06; C07D403/12; C07D405/12; C07D409/12; C07D413/14; C07D417/12
Domestic Patent References:
JP2011513245A
Foreign References:
WO1999048913A1
Attorney, Agent or Firm:
Alga Patent Office, a patent business corporation
Miyuki Ariga
Toshio Takano
Toshio Nakajima
Masaki Murata
Hiroto Yamamoto



 
Previous Patent: JPH05503556

Next Patent: JPH05503558