Title:
プロテアーゼ阻害剤および抗ウイルス剤としての5,6-ジヒドロピロン誘導体
Document Type and Number:
Japanese Patent JP3698435
Kind Code:
B2
Abstract:
The present invention relates to novel 5,6-dihydropyrone derivatives and related structures which potently inhibit the HIV aspartyl protease blocking HIV infectivity. The 5,6-dihydropyrone derivatives are useful in the development of therapies for the treatment of bacterial and viral infections and diseases, including AIDS. The present invention is also directed to methods of synthesis of multifunctionalized 5,6-dihydropyrones and of related structures.
Inventors:
Edmund Lee, Ellsworth
Lenny, Elizabeth
Tate, Bradley Dane
Lenny, Elizabeth
Tate, Bradley Dane
Application Number:
JP51445495A
Publication Date:
September 21, 2005
Filing Date:
October 26, 1994
Export Citation:
Assignee:
Park Davis and Company
International Classes:
A61K31/35; A61K31/351; A61K31/352; A61K31/365; C07D335/02; A61K31/366; A61K31/38; A61K31/382; A61K31/44; A61K31/443; A61P31/04; A61P31/12; A61P31/18; C07C321/26; C07C323/20; C07C323/22; C07C381/04; C07D211/84; C07D211/86; C07D309/32; C07D309/38; C07D311/96; C07D405/04; C07D405/06; C07D405/12; C07D407/06; C07D407/12; (IPC1-7): C07D309/32; A61K31/366; A61P31/04; A61P31/18
Domestic Patent References:
| JP53034776A | ||||
| JP58213775A |
Foreign References:
| US3931235 |
Attorney, Agent or Firm:
Chika Takagi
Tatsuo Sato
Kosuke Nishimura
Tatsuo Sato
Kosuke Nishimura
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