Title:
7-[(3-クロロ-6,11-ジヒドロ-6-メチルジベンゾ[c,f][1,2]チアゼピン-11-イル)アミノ]ヘプタン酸S,S-ジオキシドの多形相ならびにそれらの製造及び使用方法
Document Type and Number:
Japanese Patent JP2010520298
Kind Code:
A
Abstract:
Disclosed herein are novel polymorphs of 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid S,S-dioxide. Also described herein are novel pharmaceutical compositions comprising one or more 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid S,S-dioxide polymorphs, methods of making, and related methods of treatment.
Inventors:
Sanson, Machine
Application Number:
JP2009552831A
Publication Date:
June 10, 2010
Filing Date:
March 04, 2008
Export Citation:
Assignee:
Transform Pharmaceuticals Incorporated
International Classes:
C07D281/02; A61K31/554; A61P1/04; A61P11/06; A61P25/00; A61P25/14; A61P25/24
Domestic Patent References:
| JPS4941354A | 1974-04-18 | |||
| JPS62198672A | 1987-09-02 | |||
| JPH07258089A | 1995-10-09 | |||
| JP2006516643A | 2006-07-06 | |||
| JP2001504758A | 2001-04-10 | |||
| JP2004530545A | 2004-10-07 | |||
| JP2002536374A | 2002-10-29 |
Foreign References:
| US3758528A | 1973-09-11 |
Other References:
JPN6013006697; Ｄａｎｉｌｏ Ｇｉａｎｎｏｔｔｉ ｅｔ ａｌ: 'Ｎｅｗ ｄｉｂｅｎｚｏｔｈｉａｄｉａｚｅｐｉｎｅ ｄｅｒｉｖａｔｉｖｅｓ ｗｉｔｈ ａｎｔｉｄｅｐｒｅｓｓａｎｔ ａｃｔｉｖｉｔｉｅｓ' Ｊｏｕｒｎａｌ ｏｆ Ｍｅｄｉｃｉｎａｌ Ｃｈｅｍｉｓｔｒｙ Ｖｏｌ．３４， Ｎｏ．４, 1991, ｐ．１３５６-１３６２
JPN6014012260; Ｍ．Ｄ． Ｌｕｑｕｅ ｄｅ Ｃａｓｔｒｏ ｅｔ ａｌ: 'Ｕｌｔｒａｓｏｕｎｄ-ａｓｓｉｓｔｅｄ ｃｒｙｓｔａｌｌｉｚａｔｉｏｎ （ｓｏｎｏｃｒｙｓｔａｌｌｉｚａｔｉｏｎ）' Ｕｌｔｒａｓｏｎｉｃｓ Ｓｏｎｏｃｈｅｍｉｓｔｒｙ Ｖｏｌ．１４， Ｎｏ．６, 2007, ｐ．７１７-７２４
JPN6014012260; Ｍ．Ｄ． Ｌｕｑｕｅ ｄｅ Ｃａｓｔｒｏ ｅｔ ａｌ: 'Ｕｌｔｒａｓｏｕｎｄ-ａｓｓｉｓｔｅｄ ｃｒｙｓｔａｌｌｉｚａｔｉｏｎ （ｓｏｎｏｃｒｙｓｔａｌｌｉｚａｔｉｏｎ）' Ｕｌｔｒａｓｏｎｉｃｓ Ｓｏｎｏｃｈｅｍｉｓｔｒｙ Ｖｏｌ．１４， Ｎｏ．６, 2007, ｐ．７１７-７２４
Attorney, Agent or Firm:
Patent business corporation Odashima patent office