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Title:
ACYLSULFONAMIDE DERIVATIVE
Document Type and Number:
Japanese Patent JP2005119987
Kind Code:
A
Abstract:

To provide an ACC activity inhibitor which is effective for treating hyperlipemia induced by obesity and fatness, impaired glucose tolerance estimated to be based on fatty liver and insulin resistance, diabetes, diabetic complication (diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, diabetic great vessel disease), hypertension, and arteriosclerosis, and to provide a therapeutic method using the same.

This specific acylsulfonamide derivative exhibiting an ACC (acetyl CoA carboxylase) activity-inhibiting action effective for treating hyperlipemia, fatty liver, impaired glucose tolerance, diabetes, diabetic complication, hypertension, and arteriosclerosis, or its analogue or its pharmaceutically acceptable salt.


Inventors:
ICHINOSE HIDEHIRO
NIHEI YUKIO
YAMAMOTO TAKASHI
SUZUKI NOBUYASU
NAKANISHI EIJI
KONDO NOBUO
Application Number:
JP2003354530A
Publication Date:
May 12, 2005
Filing Date:
October 15, 2003
Export Citation:
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Assignee:
AJINOMOTO KK
International Classes:
C07D239/70; A61K31/352; A61K31/39; A61K31/436; A61K31/445; A61K31/527; A61K45/00; A61P1/16; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P13/12; A61P25/02; A61P27/02; A61P43/00; C07D211/30; C07D211/62; C07D311/96; C07D327/06; C07D491/107; (IPC1-7): C07D211/62; A61K31/352; A61K31/39; A61K31/436; A61K31/445; A61K31/527; A61K45/00; A61P1/16; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P13/12; A61P25/02; A61P27/02; A61P43/00; C07D211/30; C07D239/70; C07D311/96; C07D327/06; C07D491/107