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Title:
向上した水溶解度を有するアミド含有化合物およびアミド含有化合物の水溶解度を向上させる方法
Document Type and Number:
Japanese Patent JP2005520782
Kind Code:
A
Abstract:
The present invention is directed to novel amide-containing compounds which have an improved solubility and a method of improving the solubility of amide-containing compounds. The amide-containing compounds include oxazolidinone compounds and the bioavailability of these oxazolidinone compounds is improved by improving the solubility thereof.

Inventors:
Jackson Be Hester Jr.
Application Number:
JP2003512212A
Publication Date:
July 14, 2005
Filing Date:
July 12, 2002
Export Citation:
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Assignee:
Pharmacia & Up John Company LRC
International Classes:
A61K31/422; A61K31/4439; A61K31/496; A61K31/5377; A61K31/541; A61K31/55; A61K31/554; A61P25/16; A61P31/04; A61P43/00; C07D263/20; C07D405/10; C07D411/10; C07D413/04; C07D413/10; C07D263/22; C07D413/12; C07D417/10; C07D417/12; C07D417/14; C07D471/10; C07D521/00; C07F9/653; C07F9/6558; F24C15/10; (IPC1-7): C07D263/22; A61K31/422; A61K31/4439; A61K31/496; A61K31/5377; A61K31/541; A61K31/55; A61K31/554; A61P25/16; A61P31/04; A61P43/00; C07D405/10; C07D413/10; C07D413/12; C07D417/10
Attorney, Agent or Firm:
Mitsuo Tanaka
Masaki Yano