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Title:
BTK阻害剤
Document Type and Number:
Japanese Patent JP2018502159
Kind Code:
A
Abstract:
本発明は一連のBTK阻害剤を公開した。具体的には、式(I)、式(II)、式(III)又は式(IV)に示された化合物、そのその薬学的に許容される塩、その互変異性体、又はそのプロドラッグを公開した。

Inventors:
Wang Gakuhai
Wu Seitoku
Courage
Senharu
Li Liu
Kokuhei
Rakuyo
Reiken
Guo Ryosuke
Performance
Yellow Lou
Chen Akebono
To Eika
Yang Nakabun
Zhang Owen
Strength
Field flower
Flat gloss
Chen Hai Liang
Sun Bun Kiyoshi
What
Uncleanness
Yang
Calm
Weekly sentence
Stillness
Zhang Yi
Liu Chuen
Application Number:
JP2017555826A
Publication Date:
January 25, 2018
Filing Date:
June 17, 2015
Export Citation:
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Assignee:
HUBEI BIO-PHARMACEUTICAL INDUSTRIAL TECHNOLOGICAL INSTITUTE INC.
International Classes:
C07D213/74; A61K31/454; A61K31/495; A61K31/496; A61K31/497; A61K31/5025; A61K31/506; A61K31/519; A61K31/53; A61K31/5355; A61K31/5365; A61K31/55; A61K31/553; A61P43/00; C07D401/12; C07D401/14; C07D403/04; C07D455/02; C07D471/04; C07D487/04; C07D498/04
Attorney, Agent or Firm:
Hiroyuki Hashimoto
Rie Senrai