Title:
ベンズアミド誘導体
Document Type and Number:
Japanese Patent JP4625969
Kind Code:
B2
Abstract:
This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by general formula (I):wherein R1 is aryl optionally substituted with lower alkoxy, etc.,R2 is lower alkyl, etc.,R3 is hydrogen, etc.,A is NH, etc.,E isetc.,X is -CH=CH-, -CH=N-, or S, andY is a condensed heterocyclic group, etc.,and pharmaceutically acceptable salts thereof, to processes for preparation thereof and to a pharmaceutical composition comprising the same.
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Inventors:
Hiroyuki Setoi
Takehiko Okawa
Yoshimitsu Tatsuya
Hitoshi Sawada
Yuki Sawada
Teruo Oku
Takehiko Okawa
Yoshimitsu Tatsuya
Hitoshi Sawada
Yuki Sawada
Teruo Oku
Application Number:
JP52122598A
Publication Date:
February 02, 2011
Filing Date:
November 18, 1997
Export Citation:
Assignee:
Astellas Pharma Inc.
International Classes:
C07C237/42; A61K31/40; A61K31/4035; A61K31/41; A61K31/415; A61K31/4184; A61K31/422; A61K31/454; A61K31/495; A61K31/496; A61K31/498; A61K31/517; A61K31/52; A61K31/535; A61K31/5375; A61K31/5377; A61P1/08; A61P1/16; A61P3/10; A61P7/00; A61P9/00; A61P9/12; A61P13/12; A61P43/00; C07C237/44; C07D209/08; C07D209/12; C07D209/14; C07D209/34; C07D209/42; C07D209/48; C07D215/48; C07D231/56; C07D235/06; C07D235/08; C07D235/10; C07D235/12; C07D235/14; C07D235/16; C07D235/24; C07D235/26; C07D235/28; C07D235/30; C07D235/32; C07D239/88; C07D239/96; C07D241/42; C07D249/18; C07D263/10; C07D263/30; C07D263/54; C07D263/56; C07D265/32; C07D265/34; C07D295/12; C07D295/135; C07D295/18; C07D295/185; C07D401/04; C07D401/06; C07D401/12; C07D403/04; C07D403/06; C07D403/12; C07D413/12; C07D471/04; C07D473/00; C07D487/04; C07D521/00; C07F7/18
Domestic Patent References:
| JP4154765A | ||||
| JP2009143904A |
Foreign References:
| WO1995029152A1 |
Other References:
A.Varvavas et al., Anthranoyl-anthranilic acid:a template for the development of a new class of cholecystokinin receptor ligands, Pharmazie , ドイツ, 1996年10月, vol.51 no.10, 697-700
Marie-Florence Grenier-Loustalot et al., Mechanisms and Kinetics of Polymerisation of Thermoplastic Polyimides. II. Study of ”Bridged”Dianhydride/Aromatic Amine Systems, Journal of Polymer Science,Polymer Chemistry Edition, 米国, 1993年11月, vol.31,no.12, 3049-3063
Marie-Florence Grenier-Loustalot et al., Mechanisms and Kinetics of Polymerisation of Thermoplastic Polyimides. II. Study of ”Bridged”Dianhydride/Aromatic Amine Systems, Journal of Polymer Science,Polymer Chemistry Edition, 米国, 1993年11月, vol.31,no.12, 3049-3063
Attorney, Agent or Firm:
Morita Taku
Hamai Kosuke
Hamai Kosuke