BENZOTHIOPHENE, FORMULATION CONTAINING THE SAME, AND METHOD

Title:

BENZOTHIOPHENE, FORMULATION CONTAINING THE SAME, AND METHOD

Document Type and Number:

Japanese Patent JP2009019057

Kind Code:

A

Abstract:

To provide a hydrochloride of a compound represented by formula (I), in a particulate form and having a specified size range.

Pharmaceutical compositions containing a compound of formula (I) or formulated by using the compound of formula (I) are provided, and the use of such compounds for alleviating human pathologies, including osteoporosis, serum lipid lowering, and breast cancer, is provided.

Inventors:

ARBUTHNOT GORDON N
DALDER BRIAN W
HARTAUER KERRY J
LUKE WAYNE D
STRATFORD ROBERT E JR

Application Number:

JP2008227311A

Publication Date:

January 29, 2009

Filing Date:

September 04, 2008

Export Citation:

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Assignee:

LILLY CO ELI

International Classes:

A61K31/38; C07D333/56; A61K31/00; A61K31/445; A61K31/4465; A61K31/4523; A61K31/4535; A61P3/00; A61P3/06; A61P15/00; A61P15/08; A61P19/00; A61P19/10; A61P35/00; C07D333/58; A61K31/381

Domestic Patent References:

JPH07277973A	1995-10-24
JP2000507268A	2000-06-13
JPS63112519A	1988-05-17
JPH05507466A	1993-10-28

Foreign References:

DE19534744A1	1996-03-21
WO1995017382A1	1995-06-29
WO1994008709A1	1994-04-28

Other References:

JPN4007021469; ＪＪＳＨＰＶｏｌ．２４，　Ｎｏ．１１, 1988, ｐｐ．１１７５-１１８２
JPN6012014412; 橋田　充　編: 経口投与製剤の設計と評価 , 19950210, ６９-８５, 株式会社　薬業時報社
JPN6013004728; Ｍｏｄｅｒｎ　Ｐｈａｒｍａｃｅｕｔｉｃｓ , 1979, ３５９-３６５
JPN6013004731; Ｔｈｅ　Ｔｈｅｏｒｙ　ａｎｄ　ｐｒａｃｔｉｃｅ　ｏｆ　ｉｎｄｕｓｔｒｉａｌ　ｐｈａｒｍａｃｙ２ｎｄ　Ｅｄ．, 1976, ４６６-４８５
JPN6013004734; Ｐｈａｒｍａｃｅｕｔｉｃｓ：　Ｔｈｅ　ｓｃｉｅｎｃｅ　ｏｆ　ｄｏｓａｇｅ　ｆｏｒｍ　ｄｅｓｉｇｎ , 1988, ５６４-５９０

Attorney, Agent or Firm:

Kyousei Tamura
Samejima Mutsumi
Nagatoshi Shinagawa
Yasushi Morimoto

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