Title:
BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS
Document Type and Number:
Japanese Patent JP2017048198
Kind Code:
A
Abstract:
PROBLEM TO BE SOLVED: To provide compounds and methods of treating anti-inflammatory conditions.SOLUTION: A method of treating an anti-inflammatory disease comprises administering a boron-containing compound of the formula in the figure. (Ris CN, C(O)NRR, or C(O)OR; X is N, CH, or CR; Ris halogen, an alkyl group, C(O)R, C(O)OR, OR, or NRR; it is H, an alkyl group, a heteroalkyl group, or the like; R, R, Rand Rare H, alkyl, heteroalkyl, cycloalkyl, or heterocycloalkyl; and Ris H or unsubstituted alkyl.)SELECTED DRAWING: None
Inventors:
AKAMA TSUTOMU
ZHANG YONG-KANG
CHARLES Z DING
PLATTNER JACOB J
MAPLES KIRK R
FREUND YVONNE
SANDERS VIRGINIA
XIA YI
STEPHEN J BAKER
JAMES A NIEMANN
XIAOSONG LU
MARCELO SALES
RASHMI SHARMA
RAJESHWAR SINGH
ROBERT JACOBS
CHEN DAITAO
MICHAEL RICHARD KEVIN ALLEY
ZHANG YONG-KANG
CHARLES Z DING
PLATTNER JACOB J
MAPLES KIRK R
FREUND YVONNE
SANDERS VIRGINIA
XIA YI
STEPHEN J BAKER
JAMES A NIEMANN
XIAOSONG LU
MARCELO SALES
RASHMI SHARMA
RAJESHWAR SINGH
ROBERT JACOBS
CHEN DAITAO
MICHAEL RICHARD KEVIN ALLEY
Application Number:
JP2016200922A
Publication Date:
March 09, 2017
Filing Date:
October 12, 2016
Export Citation:
Assignee:
ANACOR PHARMACEUTICALS INC
International Classes:
C07F5/02; A61K33/22; A61P1/04; A61P1/16; A61P1/18; A61P3/00; A61P3/10; A61P7/06; A61P9/00; A61P9/10; A61P11/00; A61P11/06; A61P13/12; A61P17/00; A61P17/04; A61P17/06; A61P19/00; A61P19/02; A61P25/00; A61P27/02; A61P29/00; A61P31/08; A61P31/18; A61P33/06; A61P37/02; A61P37/08; A61P43/00
Domestic Patent References:
| JP5745279B2 | 2015-07-08 | |||
| JP2008535781A | 2008-09-04 |
Foreign References:
| US20070293457A1 | 2007-12-20 | |||
| US6800645B1 | 2004-10-05 | |||
| US20060222671A1 | 2006-10-05 |
Attorney, Agent or Firm:
Yoshiyuki Inaba
Toshifumi Onuki
Toshifumi Onuki