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Title:
ファルネシルトランスフェラーゼを阻害する炭素連結イミダゾールもしくはトリアゾール置換三環状キナゾリン誘導体
Document Type and Number:
Japanese Patent JP4384505
Kind Code:
B2
Abstract:
This invention comprises the novel compounds of formula (I) wherein r, s, t, R1, R2, R3, R4, R5, and R6 have defined meanings, having farnesyl transferase inhibiting activity; their preparation, compositions containing them and their use as a medicine.

Inventors:
Anjibo, Patrick Rene
Marc Gaston, Benet
Arguyon, Jean-Michel-Jacques Raymon
Application Number:
JP2003584057A
Publication Date:
December 16, 2009
Filing Date:
April 14, 2003
Export Citation:
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Assignee:
JANSSEN PHARMACEUTICA NAAMLOZE VENNOOTSCHAP
International Classes:
C07D487/04; A61K31/437; A61K31/519; A61P35/00; A61P43/00
Foreign References:
WO2000039082A1
WO1998040383A1
WO2002024682A1
Other References:
F. OERTEL,PHARMAZIE,1990年,Vol.45,No.5,p.370
Attorney, Agent or Firm:
Patent business corporation Odashima patent office



 
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