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Patent Searching and Data


Title:
カルボキサミド誘導体並びに血栓塞栓性疾患および腫瘍の処置におけるこれらの使用
Document Type and Number:
Japanese Patent JP2004515538
Kind Code:
A
Abstract:
Novel compounds of the formula I in which R1, D, E, W, X and n are as defined in claim 1, are inhibitors of coagulation factor Xa and can be employed for the prophylaxis and/or therapy of thromboembolic diseases and for the treatment of tumours.

Inventors:
Dolsh Dieter
Medellsky, Werner
Zakura Kydis, Christos
Cezanne, Petrum
Glitz, johannes
Burns, christopher
Application Number:
JP2002549632A
Publication Date:
May 27, 2004
Filing Date:
November 21, 2001
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
A61K31/17; A61K31/27; A61K31/381; A61K31/402; A61K31/405; A61K31/4172; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4412; A61K31/445; A61K31/4453; A61K31/4468; A61K31/45; A61K31/453; A61K31/4535; A61K31/4545; A61K31/495; A61K31/497; A61K31/5375; A61K31/55; A61P7/02; A61P9/00; A61P9/08; A61P9/10; A61P29/00; A61P35/00; A61P35/04; C07C271/28; C07C273/18; C07C275/28; C07C275/30; C07C303/40; C07C311/39; C07C311/46; C07C315/04; C07C317/32; C07C323/60; C07D207/27; C07D209/18; C07D209/20; C07D211/20; C07D211/26; C07D211/58; C07D211/76; C07D213/56; C07D213/64; C07D213/74; C07D213/75; C07D223/10; C07D233/54; C07D233/64; C07D241/08; C07D265/32; C07D295/135; C07D295/12; C07D295/20; C07D295/205; C07D333/24; C07D401/04; C07D401/14; C07D405/04; C07D409/12; C07D409/14; C07D417/14; C07D207/26; (IPC1-7): C07C317/32; A61K31/17; A61K31/27; A61K31/381; A61K31/402; A61K31/405; A61K31/4172; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4412; A61K31/445; A61K31/4453; A61K31/4468; A61K31/45; A61K31/453; A61K31/4535; A61K31/4545; A61K31/495; A61K31/497; A61K31/5375; A61K31/55; A61P7/02; A61P9/00; A61P9/08; A61P9/10; A61P29/00; A61P35/00; A61P35/04; C07C273/18; C07C275/28; C07C303/40; C07C311/39; C07C315/04; C07D207/27; C07D209/18; C07D211/26; C07D211/58; C07D211/76; C07D213/56; C07D213/64; C07D213/74; C07D213/75; C07D223/10; C07D233/64; C07D241/08; C07D265/32; C07D295/12; C07D295/20; C07D333/24; C07D401/04; C07D401/14; C07D405/04; C07D409/12; C07D409/14
Attorney, Agent or Firm:
Kiyoji Kuzuwa