クロモボックスタンパク質阻害剤およびその使用

Japanese Patent JP7203018

B2

Provided herein are compounds useful as inhibitors of CBX. Also described are pharmaceutical compositions and medical uses of these compounds.

Bradner, James E.
Qi, Jun
Federation, Alexander
Jacobson, Zoe
Valka, Anthony

JP2019515887A

January 12, 2023

September 25, 2017

Click for automatic bibliography generation  

Dana Farber Cancer Institute, Incorporated

C07D405/04; A61K31/427; A61K31/4375; A61K31/4439; A61K31/4545; A61K31/47; A61K31/4709; A61K31/495; A61K31/496; A61K31/506; A61K31/5377; A61K31/541; A61K31/55; A61P35/00; A61P35/02; A61P43/00; C07D213/30; C07D213/82; C07D277/28; C07D277/48; C07D277/50; C07D277/54; C07D277/82; C07D279/12; C07D295/192; C07D401/04; C07D401/06; C07D401/12; C07D405/14; C07D417/12; C07D471/04; C07D513/18

JP2016519091A
JP2008517061A

WO2012122370A2
WO2016077632A2
WO2008154207A1
WO2010004761A1
WO2010151799A2
WO2013074059A2
WO2006094237A2
US8846320
WO2016004035A1
WO2014113467A1

ACS Medicinal Chemistry Letters,2010年07月13日,Vol.1,No.8,p371-375,doi:10.1021/ml1000273
Journal of Medicinal Chemistry,2010年02月25日,Vol.53,No.4,p1483-1495,doi:10.1021/jm900776m
ChemMedChem,2009年12月,Vol.4,No.12,p2060-2069,doi:10.1002/cmdc.200900262
RN 1624164-86-8 REGISTRYY,DATABASE REGISTRY [ONLINE],Retrieved from STN,検索日: 26 MAY 2021,2014年09月22日
RN 730948-00-2 REGISTRY,DATABASE REGISTRY [ONLINE],Retrieved from STN,検索日: 26 MAY 2021,2004年08月23日
RN 400011-90-7 REGISTRY,DATABASE REGISTRY [ONLINE],Retrieved from STN,検索日: 6 MAY 2022,2002年03月11日

Shusaku Yamamoto
Morishita Natsuki
Takatoshi Iida
Daisuke Ishikawa
Kensaku Yamamoto

Previous Patent: How to detect lentivirus

Next Patent: METHOD OF DETERMINING FUNCTION OF PUSHBUTTON SWITCH AND ASSEMBLY THEREFOR