Title:
活性剤デリバリーのための化合物及び組成物
Document Type and Number:
Japanese Patent JP4637365
Kind Code:
B2
Abstract:
Compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well.
Inventors:
Pinwa Tan
Andrea Leone-Bay
David Gschneider
Eugene N Ballantosevic
Andrea Leone-Bay
David Gschneider
Eugene N Ballantosevic
Application Number:
JP2000600970A
Publication Date:
February 23, 2011
Filing Date:
February 25, 2000
Export Citation:
Assignee:
Emisfair Technologies Inc.
International Classes:
C07C235/60; A61K9/00; A61K9/08; A61K9/14; A61K9/20; A61K9/48; A61K31/4015; A61K31/70; A61K31/715; A61K31/726; A61K38/00; A61K38/22; A61K38/27; A61K45/06; A61K47/04; A61K47/10; A61K47/16; A61K47/18; A61K47/22; A61P5/06; A61P5/18; A61P7/02; A61P43/00; C07D207/27; C07D233/61; C07D295/12; C07D295/13; C07D521/00; C07D207/26
Domestic Patent References:
| JP5239005A |
Foreign References:
| US2810718 |
Other References:
Davaran, Soodabeh; Hanaee, Jalal; Khosravi, Abbas,Release of 5-aminosalicylic acid from acrylic type polymeric prodrugs designed for colon-specific drug delivery,Journal of Controlled Release,1999年,58(3),279-287
Johansen, Marianne; Bundgaard, Hans,Pro-drugs as drug delivery systems. XIII. Kinetics of decomposition of N-Mannich bases of salicylamide and assessment of their suitability as possible pro-drugs for amines,International Journal of Pharmaceutics,1980年,7(2),119-127
Phillips, Barrie Maurice; Havera, Herbert J.; Hammes, Toni L.,Ring opening of cyclic salicylamides,Journal of Pharmaceutical Sciences,1969年,58(11),1414-1416
Jaszay, Zsuzsa M.; Petnehazy, Imre; Toke, Laszlo,Phase-transfer catalyzed synthesis of amides and esters of carboxylic acids,Synthesis,1989年,(10),745-747
Minasyan, S. A.; Arakelyan, E. A.; Pogosyan, A. V.; Markaryan, E. A.,Phenolic acid derivatives. XXXIII. Synthesis of (dialkylamino)alkylamides of phenolic acids,Armyanskii Khimicheskii Zhurnal,1986年,39(3),169-174
Bahekar, Rajesh H.; Gaikwad, N. J.,Synthesis and biological evaluation of indomethacin conjugates with salicylamide and its Mannich bases: a mutual prodrug approach,Indian Drugs,1998年,35(10),648-652
Ottenbrite, Raphael M.; Hu, Bin,Synthesis and characterization of PEG-EDTA bidentates as oral drug systems,Polymer Preprints (American Chemical Society, Division of Polymer Chemistry),2000年,41(1),6-7
Levant, Beth; Moehlenkamp, Jeffrey D.; Morgan, Kimberly a.; Leonard, Neda L.; Cheng, C. C.,Modulation of [3H]quinpirole binding in brain by monoamine oxidase inhibitors: evidence for a potential novel binding site,Journal of Pharmacology and Experimental Therapeutics,1996年,278(1),145-153
Johansen, Marianne; Bundgaard, Hans,Pro-drugs as drug delivery systems. XIII. Kinetics of decomposition of N-Mannich bases of salicylamide and assessment of their suitability as possible pro-drugs for amines,International Journal of Pharmaceutics,1980年,7(2),119-127
Phillips, Barrie Maurice; Havera, Herbert J.; Hammes, Toni L.,Ring opening of cyclic salicylamides,Journal of Pharmaceutical Sciences,1969年,58(11),1414-1416
Jaszay, Zsuzsa M.; Petnehazy, Imre; Toke, Laszlo,Phase-transfer catalyzed synthesis of amides and esters of carboxylic acids,Synthesis,1989年,(10),745-747
Minasyan, S. A.; Arakelyan, E. A.; Pogosyan, A. V.; Markaryan, E. A.,Phenolic acid derivatives. XXXIII. Synthesis of (dialkylamino)alkylamides of phenolic acids,Armyanskii Khimicheskii Zhurnal,1986年,39(3),169-174
Bahekar, Rajesh H.; Gaikwad, N. J.,Synthesis and biological evaluation of indomethacin conjugates with salicylamide and its Mannich bases: a mutual prodrug approach,Indian Drugs,1998年,35(10),648-652
Ottenbrite, Raphael M.; Hu, Bin,Synthesis and characterization of PEG-EDTA bidentates as oral drug systems,Polymer Preprints (American Chemical Society, Division of Polymer Chemistry),2000年,41(1),6-7
Levant, Beth; Moehlenkamp, Jeffrey D.; Morgan, Kimberly a.; Leonard, Neda L.; Cheng, C. C.,Modulation of [3H]quinpirole binding in brain by monoamine oxidase inhibitors: evidence for a potential novel binding site,Journal of Pharmacology and Experimental Therapeutics,1996年,278(1),145-153
Attorney, Agent or Firm:
Masatake Shiga
Tadashi Takahashi
Takashi Watanabe
Masakazu Aoyama
Suzuki Mitsuyoshi
Kazuya Nishi
Yasuhiko Murayama
Shinya Mitsuhiro
Tadashi Takahashi
Takashi Watanabe
Masakazu Aoyama
Suzuki Mitsuyoshi
Kazuya Nishi
Yasuhiko Murayama
Shinya Mitsuhiro