Title:
インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用な化合物
Document Type and Number:
Japanese Patent JP2020506895
Kind Code:
A
Abstract:
インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用である式(VII)の化合物が提供されている。薬学組成物、前記化合物を含むキット、ならびに、前記化合物に係る方法および使用もまた提供されている。
Inventors:
Richard Tea. Lewis
Matthew Hamilton
Philip Jones
Alessia Petrocchi
Naphthali Reina
Jason cross
Michelle Han
Michael soss
Timothy Makafuth
Martin Trenbrae
Matthew Hamilton
Philip Jones
Alessia Petrocchi
Naphthali Reina
Jason cross
Michelle Han
Michael soss
Timothy Makafuth
Martin Trenbrae
Application Number:
JP2019538180A
Publication Date:
March 05, 2020
Filing Date:
January 16, 2018
Export Citation:
Assignee:
BOARD OF REGENTS,THE UNIVERSITY OF TEXAS SYSTEM
International Classes:
C07C233/70; A61K31/166; A61K31/18; A61K31/192; A61K31/195; A61K31/196; A61K31/198; A61K31/216; A61K31/225; A61K31/275; A61K31/351; A61K31/4015; A61K31/4035; A61K31/404; A61K31/415; A61K31/416; A61K31/4184; A61K31/4192; A61K31/4196; A61K31/421; A61K31/437; A61K31/4375; A61K31/44; A61K31/4402; A61K31/455; A61K31/47; A61K31/4709; A61K31/4965; A61K31/50; A61K31/502; A61K31/517; A61K31/5375; A61K45/00; A61P1/04; A61P9/00; A61P19/02; A61P25/00; A61P25/14; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P27/02; A61P27/12; A61P29/00; A61P31/00; A61P31/04; A61P31/16; A61P31/18; A61P35/00; A61P35/02; A61P35/04; A61P37/06; A61P43/00; C07C233/65; C07C233/79; C07C233/84; C07C233/87; C07C235/34; C07C247/14; C07C255/44; C07C255/57; C07C255/58; C07C311/07; C07C311/14; C07C311/20; C07D207/408; C07D209/08; C07D209/34; C07D209/38; C07D209/46; C07D209/48; C07D213/64; C07D213/65; C07D213/68; C07D213/74; C07D213/75; C07D213/81; C07D213/82; C07D215/20; C07D215/22; C07D215/233; C07D215/26; C07D215/48; C07D231/12; C07D231/14; C07D231/56; C07D235/04; C07D235/26; C07D237/24; C07D237/28; C07D237/32; C07D239/28; C07D239/34; C07D239/74; C07D239/88; C07D239/94; C07D241/24; C07D249/04; C07D249/08; C07D249/18; C07D263/20; C07D295/135; C07D295/205; C07D309/04; C07D309/12; C07D401/04; C07D403/04; C07D403/06; C07D405/04; C07D413/08; C07D471/04
Domestic Patent References:
JPS559074A | 1980-01-22 | |||
JP2005535655A | 2005-11-24 | |||
JP2007531754A | 2007-11-08 |
Foreign References:
WO2016073774A2 | 2016-05-12 | |||
WO2016073738A2 | 2016-05-12 | |||
WO2016073770A1 | 2016-05-12 | |||
WO2016161960A1 | 2016-10-13 |
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Attorney, Agent or Firm:
Murai Koji
Horikawa Kaori
Horikawa Kaori