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Title:
インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用な化合物
Document Type and Number:
Japanese Patent JP2020506895
Kind Code:
A
Abstract:
インドールアミン2,3−ジオキシゲナーゼおよび/またはトリプトファンジオキシゲナーゼの阻害剤として有用である式(VII)の化合物が提供されている。薬学組成物、前記化合物を含むキット、ならびに、前記化合物に係る方法および使用もまた提供されている。

Inventors:
Richard Tea. Lewis
Matthew Hamilton
Philip Jones
Alessia Petrocchi
Naphthali Reina
Jason cross
Michelle Han
Michael soss
Timothy Makafuth
Martin Trenbrae
Application Number:
JP2019538180A
Publication Date:
March 05, 2020
Filing Date:
January 16, 2018
Export Citation:
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Assignee:
BOARD OF REGENTS,THE UNIVERSITY OF TEXAS SYSTEM
International Classes:
C07C233/70; A61K31/166; A61K31/18; A61K31/192; A61K31/195; A61K31/196; A61K31/198; A61K31/216; A61K31/225; A61K31/275; A61K31/351; A61K31/4015; A61K31/4035; A61K31/404; A61K31/415; A61K31/416; A61K31/4184; A61K31/4192; A61K31/4196; A61K31/421; A61K31/437; A61K31/4375; A61K31/44; A61K31/4402; A61K31/455; A61K31/47; A61K31/4709; A61K31/4965; A61K31/50; A61K31/502; A61K31/517; A61K31/5375; A61K45/00; A61P1/04; A61P9/00; A61P19/02; A61P25/00; A61P25/14; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P27/02; A61P27/12; A61P29/00; A61P31/00; A61P31/04; A61P31/16; A61P31/18; A61P35/00; A61P35/02; A61P35/04; A61P37/06; A61P43/00; C07C233/65; C07C233/79; C07C233/84; C07C233/87; C07C235/34; C07C247/14; C07C255/44; C07C255/57; C07C255/58; C07C311/07; C07C311/14; C07C311/20; C07D207/408; C07D209/08; C07D209/34; C07D209/38; C07D209/46; C07D209/48; C07D213/64; C07D213/65; C07D213/68; C07D213/74; C07D213/75; C07D213/81; C07D213/82; C07D215/20; C07D215/22; C07D215/233; C07D215/26; C07D215/48; C07D231/12; C07D231/14; C07D231/56; C07D235/04; C07D235/26; C07D237/24; C07D237/28; C07D237/32; C07D239/28; C07D239/34; C07D239/74; C07D239/88; C07D239/94; C07D241/24; C07D249/04; C07D249/08; C07D249/18; C07D263/20; C07D295/135; C07D295/205; C07D309/04; C07D309/12; C07D401/04; C07D403/04; C07D403/06; C07D405/04; C07D413/08; C07D471/04
Domestic Patent References:
JPS559074A1980-01-22
JP2005535655A2005-11-24
JP2007531754A2007-11-08
Foreign References:
WO2016073774A22016-05-12
WO2016073738A22016-05-12
WO2016073770A12016-05-12
WO2016161960A12016-10-13
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Attorney, Agent or Firm:
Murai Koji
Horikawa Kaori