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Title:
N-(4,5-ビスメタンスルホニル-2-メチルベンゾイル)グアニジン塩酸塩およびN-(4,5-ビスメタンスルホニル-2-メチルベンゾイル)グアニジン塩の結晶変態
Document Type and Number:
Japanese Patent JP7050005
Kind Code:
B2
Abstract:
The present invention relates to novel crystalline modifications of N-(4,5-bismethanesulfonyl-2-methylbenzoyl)guanidine hydrochloride, novel N-(4,5-bismethanesulfonyl-2-methylbenzoyl)guanidine salts and their crystalline modifications and processes of manufacturing and pharmaceutical formulations thereof.

Inventors:
Becker, accelerator
Gallon, gilmarie
Saar, christophe
Cune, clemens
Application Number:
JP2018560718A
Publication Date:
April 07, 2022
Filing Date:
January 27, 2017
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
C07C317/44; A61K31/155; A61P3/04; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P13/12; A61P21/00; A61P25/00; A61P35/00; A61P43/00; C07C315/06
Domestic Patent References:
JP2003512451A
JP2011519877A
JP9052876A
Other References:
平山令明編,有機化合物結晶作製ハンドブック -原理とノウハウ-,丸善株式会社,2008年07月25日,p.57-84
Journal of Pharmaceutical Sciences,1977年,Vol.66, No.1,p.1-19
Attorney, Agent or Firm:
Kiyokazu