Title:
Crystalline solvent Hydrate and the complex of a *1 which has amino acid as SGLT2 diabetic inhibitor for medical treatment (1S), and 5* anhydro *1*C* (3* (phenyl) (methyl) phenyl) *D* guru Shitoru derivative
Document Type and Number:
Japanese Patent JP5937187
Kind Code:
B2
Abstract:
The present invention relates to a pharmaceutical composition comprising a therapeutically effective amount of a crystalline (2S,3R,4S,5S,6R)-2-[4-chloro-3-(4-ethoxy-benzyl)-phenyl] -6-hydroxymethyl-2-methoxy-tetrahydro-pyran-3,4,5-triol (S)-propylene glycol solvate (compound Ia) as SGLT2 inhibitor for treating diabetes.
Inventors:
Jack Z Googoustus
Hildegard Robbinger
Srivilla Ramakrishnan
Prashant Pee Deshpande
Jeffrey T. Bean
Chiagen Rye
Chen Wan
Peter Liebel
John Anthony Grosso
Alexandra A. Nursle
Janak Shin
John Di Dimarco
Hildegard Robbinger
Srivilla Ramakrishnan
Prashant Pee Deshpande
Jeffrey T. Bean
Chiagen Rye
Chen Wan
Peter Liebel
John Anthony Grosso
Alexandra A. Nursle
Janak Shin
John Di Dimarco
Application Number:
JP2014250141A
Publication Date:
June 22, 2016
Filing Date:
December 10, 2014
Export Citation:
Assignee:
ASTRAZENECA AKTIEBOLAG
International Classes:
C07H7/04
Foreign References:
| WO2004063209A2 |
Other References:
化学実験操作法 上巻,1963年,pp.371-399
Attorney, Agent or Firm:
Samejima Mutsumi
Nagatoshi Shinagawa
Yasushi Morimoto
Nagatoshi Shinagawa
Yasushi Morimoto