Title:
KEAP1のモジュレーターとしての環状シアノエノン誘導体
Document Type and Number:
Japanese Patent JP2023535323
Kind Code:
A
Abstract:
本発明は、式(I)〔式中、R1、R2、R3、R4及びmは、本明細書中で定義されているとおりである〕で表される環状シアノエノン誘導体又はその薬学的に許容される塩若しくは溶媒和物に関する。本発明は、さらに、式(I)で表される環状シアノエノン誘導体を含んでいる医薬組成物及び治療におけるそれらの使用にも関する。【化1】TIFF2023535323000310.tif44169
Inventors:
Altman, michael
Candito, David A
Christian, Alec Aich
DiPietro, Ornella
Lou, Min
Liu Pin
Mansour, Umal Falk
Many, Katrina Marie
Musacchio, Andrew Jay
Parani, Anandang
Reuters Shan, Michael H
Shaw, David Matthew
St-Galle, Stephen
Candito, David A
Christian, Alec Aich
DiPietro, Ornella
Lou, Min
Liu Pin
Mansour, Umal Falk
Many, Katrina Marie
Musacchio, Andrew Jay
Parani, Anandang
Reuters Shan, Michael H
Shaw, David Matthew
St-Galle, Stephen
Application Number:
JP2023501769A
Publication Date:
August 17, 2023
Filing Date:
July 15, 2021
Export Citation:
Assignee:
Merck Sharp & Dome LLC
International Classes:
C07C255/46; A61K31/122; A61K31/136; A61K31/16; A61K31/166; A61K31/18; A61K31/337; A61K31/341; A61K31/343; A61K31/352; A61K31/381; A61K31/397; A61K31/4025; A61K31/403; A61K31/4155; A61K31/4188; A61K31/4192; A61K31/42; A61K31/422; A61K31/4245; A61K31/428; A61K31/433; A61K31/4355; A61K31/438; A61K31/44; A61K31/4427; A61K31/4439; A61K31/4709; A61K31/497; A61K31/501; A61K31/506; A61K31/5377; A61K31/5386; A61P21/00; A61P25/00; A61P25/02; A61P25/14; A61P25/16; A61P25/28; A61P27/16; C07D205/12; C07D209/54; C07D209/96; C07D213/81; C07D213/82; C07D221/20; C07D261/18; C07D265/36; C07D271/06; C07D305/14; C07D307/94; C07D311/96; C07D333/24; C07D401/04; C07D401/06; C07D401/14; C07D403/04; C07D403/06; C07D403/10; C07D407/04; C07D407/06; C07D409/08; C07D409/10; C07D413/04; C07D413/06; C07D413/10; C07D413/14; C07D417/06; C07D417/10; C07D471/04; C07D487/04; C07D491/048; C07D495/04; C07D498/04
Attorney, Agent or Firm:
Makoto Ono
Kennori Kanayama
Yoshiyuki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Yoshie Sakurada
Yosuke Kawasaki
Youichi Iino
Yusuke Ichikawa
Sohei Aya
Takahiro Suzuki
Yoshikazu Iwase
Yasufumi Shiroyama
Kennori Kanayama
Yoshiyuki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Yoshie Sakurada
Yosuke Kawasaki
Youichi Iino
Yusuke Ichikawa
Sohei Aya
Takahiro Suzuki
Yoshikazu Iwase
Yasufumi Shiroyama