Title:
タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
Document Type and Number:
Japanese Patent JP6490713
Kind Code:
B2
Abstract:
The present invention relates to certain diaryl macrocyclic compounds, pharmaceutical compositions containing them, and methods of using them, including methods for treating cancer, pain, neurological diseases, autoimmune diseases, and inflammation.
Inventors:
Jinron Gene Tsui
Eshan lee
Evan W. Rogers
Dayon Jai
Eshan lee
Evan W. Rogers
Dayon Jai
Application Number:
JP2016566857A
Publication Date:
March 27, 2019
Filing Date:
January 23, 2015
Export Citation:
Assignee:
TP THERAPEUTICS,INC.
International Classes:
C07D498/16; A61K31/519; A61P25/00; A61P25/04; A61P29/00; A61P37/06; A61P43/00; C07D498/22; C07D515/16
Domestic Patent References:
JP2013530142A | ||||
JP2012502043A |
Foreign References:
WO2013134219A1 | ||||
WO2013001310A1 |
Other References:
J. Am. Chem. Soc.,1961年,83,635-642
Tetrahedron Letters,2005年,46,3007-3010
ACS Medicinal Chemistry Letters,2014年 1月10日,5,193-198
Tetrahedron Letters,2005年,46,3007-3010
ACS Medicinal Chemistry Letters,2014年 1月10日,5,193-198
Attorney, Agent or Firm:
Takuji Yamada
Aoyama Aoi
Michiko Matsutani
Yasushi Ochiai
Aoyama Aoi
Michiko Matsutani
Yasushi Ochiai
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