Title:
グルココルチコイド受容体モジュレーター
Document Type and Number:
Japanese Patent JP4815566
Kind Code:
B2
Abstract:
The present invention provides non-steroidal compounds of formula I which are selective modulators (i.e., agonist and antagonists) of a steroid receptor, specifically, the glucocorticoid receptor. The present invention also provides pharmaceutical compositions containing these compounds and methods for using these compounds to treat animals requiring glucocorticoid receptor agonist or antagonist therapy. Glucocorticoid receptor modulators are useful to treat diseases, such as obesity, diabetes, inflammation and others as described below. The present invention also provides intermediates and processes for preparing these compounds
Inventors:
Dow, Robert Lee
Ryu, Kevin Khun-Chin
Bradley Paul, Morgan
Andrew Gordon, Swick
Ryu, Kevin Khun-Chin
Bradley Paul, Morgan
Andrew Gordon, Swick
Application Number:
JP2006157094A
Publication Date:
November 16, 2011
Filing Date:
June 06, 2006
Export Citation:
Assignee:
Pfizer Products Inc.
International Classes:
C07C39/23; A61K31/045; C07D295/12; A61K31/047; A61K31/05; A61K31/06; A61K31/11; A61K31/122; A61K31/133; A61K31/136; A61K31/137; A61K31/15; A61K31/166; A61K31/19; A61K31/192; A61K31/215; A61K31/255; A61K31/27; A61K31/275; A61K31/325; A61K31/336; A61K31/341; A61K31/351; A61K31/357; A61K31/365; A61K31/381; A61K31/40; A61K31/41; A61K31/4164; A61K31/4196; A61K31/4245; A61K31/425; A61K31/426; A61K31/428; A61K31/433; A61K31/4375; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/445; A61K31/4453; A61K31/451; A61K31/4535; A61K31/495; A61K31/496; A61K31/4965; A61K31/517; A61K31/5375; A61K31/5377; A61K45/00; A61P3/04; A61P3/10; A61P5/14; A61P5/44; A61P11/02; A61P11/06; A61P19/02; A61P25/00; A61P25/22; A61P25/24; A61P25/28; A61P27/16; A61P29/00; A61P37/02; A61P43/00; C07C35/42; C07C49/675; C07C49/737; C07C49/747; C07C49/755; C07C49/757; C07C65/17; C07C69/00; C07C215/50; C07C215/74; C07C225/22; C07C233/58; C07C235/48; C07C235/66; C07C247/24; C07C251/44; C07C251/52; C07C251/60; C07C255/53; C07C255/54; C07C271/10; C07C271/44; C07C271/52; C07C281/04; C07C307/02; C07C309/65; C07C309/66; C07C309/73; C07C311/04; C07C311/08; C07C311/51; C07C317/18; C07C333/04; C07D207/09; C07D211/22; C07D211/46; C07D213/22; C07D213/30; C07D213/40; C07D213/75; C07D231/40; C07D231/56; C07D233/61; C07D239/26; C07D239/34; C07D241/12; C07D241/18; C07D241/20; C07D249/08; C07D249/14; C07D257/04; C07D271/06; C07D271/07; C07D277/24; C07D277/28; C07D277/56; C07D295/08; C07D295/092; C07D295/13; C07D295/185; C07D295/205; C07D303/14; C07D317/36; C07D333/16; C07D401/04; C07D413/04; C07D413/06; C07D455/06
Domestic Patent References:
| JP5502462A | ||||
| JP62056422A | ||||
| JP61271216A | ||||
| JP43000505B1 |
Other References:
Int. J. Biochem.,1989年,21(5),p.463-468
Attorney, Agent or Firm:
Yoshinobu Murofushi
High Hoji Koji
Junko Miyazawa
Noh four
High Hoji Koji
Junko Miyazawa
Noh four