Title:
HIVウイルス侵入阻害剤
Document Type and Number:
Japanese Patent JP4823063
Kind Code:
B2
Abstract:
The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with other anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS.
Inventors:
Van Aker, Kenrath Rodebijk August
Wiegerink, Piet Tom Bale Paul
Michelle, Reve Emma Jean
Thali, Abdela
Wiegerink, Piet Tom Bale Paul
Michelle, Reve Emma Jean
Thali, Abdela
Application Number:
JP2006525834A
Publication Date:
November 24, 2011
Filing Date:
September 10, 2004
Export Citation:
Assignee:
Tabebotech Pharmaceuticals Limited
International Classes:
C07C233/29; A61K31/167; A61K31/18; A61K31/194; A61K31/198; A61K31/222; A61K31/235; A61K31/341; A61K31/36; A61K31/40; A61K31/47; A61K31/4709; A61K31/472; A61K31/495; A61P31/18; C07C233/73; C07C233/75; C07C235/16; C07C235/24; C07C235/56; C07C237/04; C07C311/21; C07C311/29; C07D207/06; C07D215/08; C07D215/26; C07D217/02; C07D295/12; C07D295/13; C07D295/14; C07D295/15; C07D307/56; C07D307/68; C07D317/68; C07D405/12; C07D405/14
Domestic Patent References:
| JPH036527A | 1991-01-14 | |||
| JPH07164756A | 1995-06-27 | |||
| JPH11277906A | 1999-10-12 | |||
| JPH06181264A | 1994-06-28 | |||
| JPS5176232A | 1976-07-01 | |||
| JPS49128933A | 1974-12-10 | |||
| JP2001329053A | 2001-11-27 | |||
| JP2001519808A | 2001-10-23 | |||
| JP2001515470A | 2001-09-18 | |||
| JP2002502850A | 2002-01-29 |
Foreign References:
| WO2000013058A1 | 2000-03-09 | |||
| US5070096A | 1991-12-03 |
Attorney, Agent or Firm:
Patent business corporation Odashima patent office