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Title:
複素環式アペリン受容体(APJ)アゴニスト及びそれらの使用
Document Type and Number:
Japanese Patent JP7104690
Kind Code:
B2
Abstract:
This disclosure is directed to agonists of the apelin receptor (APJ) with heterocyclic cores and uses of such agonists.

Inventors:
Scott Pea Lanyon
Langan Maitra
Sanjunarayanan
Kenneth S Leader
Application Number:
JP2019508240A
Publication Date:
July 21, 2022
Filing Date:
October 11, 2017
Export Citation:
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Assignee:
Research Triangle Institute
International Classes:
C07D249/10; A61K31/4196; A61K31/4439; A61K31/454; A61K31/4545; A61K31/506; A61K45/00; A61P1/16; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P7/02; A61P9/00; A61P9/12; A61P11/06; A61P13/12; A61P25/00; A61P29/00; A61P35/00; A61P43/00; C07D401/04; C07D401/12; C07D401/14; C07D403/12; C07D417/14
Domestic Patent References:
JP2005504805A
JP2006501275A
JP2005508384A
JP2014525912A
JP2015524449A
JP2015521193A
JP2010500336A
JP2010518110A
JP58194866A
JP59098004A
JP2009529540A
JP2017523126A
JP2019501899A
Foreign References:
WO2014053533A1
WO2011005052A2
WO2006043594A1
WO2011156557A2
WO2015184011A2
Other References:
DYCK, Brian,Bioorganic & Medicinal Chemistry Letters,2004年,14,1151-1154
CHO, Kyoung-in,ACS Chemical Neuroscience,2015年,6,1476-1485
STN International,1938533-13-1, 1938292-99-9, 1831835-31-4, 1830232-36-4ほか,File REGISTRY [online],2016年06月24日
HERSHBERGER, Paul M.,Bioorganic & Medicinal Chemistry Letters,2014年,24,262-267
NARAYANAN, Sanju,Bioorganic & Medicinal Chemistry,2016年,24,3758-3770
Attorney, Agent or Firm:
Kenji Sugimura
Mitsutsugu Sugimura
Mutsumi Yamamoto