Title:
脱ハロゲン化なしにハロゲノアルケンを水素化する方法
Document Type and Number:
Japanese Patent JP2012530116
Kind Code:
A
Abstract:
A process for producing bortezomib N-(pyrazin-2-yl)carbonyl-L-phenylalanine-L-leucine boronic acid) comprising the step of deprotecting the compound of formula XII: to yield bortezomib.
Inventors:
Gazuitsuchi Smirobich, Ivana
Casal, Zenko
Casal, Zenko
Application Number:
JP2012515516A
Publication Date:
November 29, 2012
Filing Date:
June 18, 2010
Export Citation:
Assignee:
Let's Farmer's Medicals Day Day
International Classes:
C07F5/04; B01J31/22; B01J31/24; C07B31/00; C07B53/00; C07B57/00; C07B61/00
Domestic Patent References:
| JP2012530115A | 2012-11-29 | |||
| JPH08259477A | 1996-10-08 | |||
| JPH0769943A | 1995-03-14 |
Foreign References:
| WO2002045834A2 | 2002-06-13 |
Attorney, Agent or Firm:
Kawaguchi International Patent Office
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