【発明の名称】モチリン受容体のアンタゴニストとして有用なシクロペンテン誘導体

Title:

【発明の名称】モチリン受容体のアンタゴニストとして有用なシクロペンテン誘導体

Document Type and Number:

Japanese Patent JP2001521030

Kind Code:

A

Abstract:

The compounds of formula I are useful in treating gastrointestinal disorders associated with antagonizing the motilin receptor disorders. The compounds compete with erythromycin and motilin for the motilin receptor. In addition the compounds are antagonists of the contractile smooth muscle response to those ligands.

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Inventors:

Robert H. Chain
Sheung, Min
Moore, Jiyon Bee, Giunia
Beavers, Mary Pat

Application Number:

JP2000517958A

Publication Date:

November 06, 2001

Filing Date:

October 27, 1998

Export Citation:

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Assignee:

Ortho-McNeill Pharmacy Incorporated

International Classes:

A61K31/16; A61K31/167; A61K31/216; A61K31/40; A61K31/4409; A61K31/445; A61K31/4468; A61K31/5375; A61K31/5377; A61P1/00; A61P1/06; A61P1/12; A61P43/00; C07C233/41; C07C233/78; C07C323/36; C07C323/42; C07D211/26; C07D211/58; C07D213/81; C07D295/08; C07D295/092; C07D295/13; C07D295/22; C07D295/24; C07D317/68; C07D333/38; (IPC1-7): C07C233/41; A61K31/16; A61K31/167; A61K31/216; A61K31/40; A61K31/445; A61K31/5375; A61K31/5377; A61P1/00; A61P1/06; A61P1/12; A61P43/00; C07C233/78; C07C323/36; C07C323/42; C07D211/58; C07D213/81; C07D295/08; C07D295/22; C07D317/68

Attorney, Agent or Firm:

Heiyoshi Odashima

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