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Patent Searching and Data


Title:
AKT活性の阻害剤
Document Type and Number:
Japanese Patent JP5923043
Kind Code:
B2
Abstract:
The invention relates to a series of compounds with particular activity as inhibitors of the serine-threonine kinase AKT. Also provided are pharmaceutical compositions comprising same as well as methods for treating cancer.

Inventors:
Zan, Rixin
Trevit, Graham, Peter
Meal, Hugoose
Frank, Barkamp
Harrison, Timothy
Wilkinson, Andrew, John
Fabricius, Charles-Henri
Application Number:
JP2012545434A
Publication Date:
May 24, 2016
Filing Date:
December 23, 2010
Export Citation:
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Assignee:
Almac Discovery Limited
International Classes:
C07D215/20; A61K31/436; A61K31/437; A61K31/444; A61K31/47; A61K31/4745; A61K31/4985; A61K31/519; A61K31/5377; A61K31/5383; A61K31/542; A61K31/546; A61K31/551; A61K31/553; A61K41/00; A61P35/00; A61P35/02; A61P43/00; C07D215/38; C07D471/04; C07D491/052; C07D491/147; C07D498/04; C07D515/04
Domestic Patent References:
JP2009501698A
JP2007524710A
Foreign References:
WO2009148916A1
WO2008011032A1
Attorney, Agent or Firm:
Yusuke Hiraki
Satoshi Fujita
Eiichi Arai
Natsuo Tanaka