Title:
INHIBITOR FOR CYTOCHROME P450 MONOOXYGENASE AND INTERMEDIATE RELATED THERETO
Document Type and Number:
Japanese Patent JP2018162274
Kind Code:
A
Abstract:
PROBLEM TO BE SOLVED: To provide an inhibitor for cytochrome P450 monooxygenase and a synthetic intermediate thereof.SOLUTION: Using a compound of formula IV as a raw material, a compound of formula I and a salt thereof are prepared through a multistage reaction.SELECTED DRAWING: None
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Inventors:
RICHARD POLNIASZEK
PFEIFFER STEVEN
RICHARD YU
AARON CULLEN
ERIC DOWDY
DUONG TRAN
KENT KENNETH
ZHOU ZHONGXIN
DOUG CORDEAU
LEAH EASTON
PFEIFFER STEVEN
RICHARD YU
AARON CULLEN
ERIC DOWDY
DUONG TRAN
KENT KENNETH
ZHOU ZHONGXIN
DOUG CORDEAU
LEAH EASTON
Application Number:
JP2018115527A
Publication Date:
October 18, 2018
Filing Date:
June 18, 2018
Export Citation:
Assignee:
GILEAD SCIENCES INC
International Classes:
C07C307/06; A61K31/5377; A61P43/00; C07C211/27; C07C303/34; C07D203/24; C07D277/28; C07D417/12
Attorney, Agent or Firm:
Hidesaku Yamamoto
Natsuki Morishita
Natsuki Morishita