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Title:
カリケアマイシン誘導体を合成するための中間体および方法
Document Type and Number:
Japanese Patent JP6494240
Kind Code:
B2
Abstract:
and to methods of synthesizing and purifying calicheamicin derivatives.

Inventors:
Robert Wayne Dagger
Rio Joseph Retendure
Vimarkumar Babab Hai Patel
Amanaus Chassetree Prashad
Chung Chung Chung Chung
Application Number:
JP2014218815A
Publication Date:
April 03, 2019
Filing Date:
October 28, 2014
Export Citation:
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Assignee:
Pfizer Inc.
International Classes:
C07C323/52; C07C319/06; C07C319/20; C07D207/46; C07H15/26
Domestic Patent References:
JP2009527557A
JP2010528031A
JP2007210974A
JP2005524700A
JP2096599A
JP8048637A
Foreign References:
WO2007014054A2
WO2008032164A2
Other References:
Theodora W. Greene 他,Protective Groups in Organic Synthesis,米国,John Wiley & Sons, Inc.,1999年,3rd ed.,P454-466
Ricart, A. ,Antibody-Drug Conjugates of Calicheamicin Derivative: Gemtuzumab Ozogamicin and Inotuzumab Ozogamicin,Clin Cancer Res ,2011年,17(20),6417-6427
Attorney, Agent or Firm:
Noh four
Junko Miyazawa
Maki Sato
Tatsuta Miyuki