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Title:
アセトアミド誘導体並びに凝固第Xaおよび第VIIa因子の阻害剤としてのその使用
Document Type and Number:
Japanese Patent JP2004505106
Kind Code:
A
Abstract:
Novel compounds of the formula I, in which R, R<1 >and R<2 >are as defined in patent claim 1, are inhibitors of coagulation factor Xa and VIIa and can be employed for the treatment of thromboses, myocardial infarction, arteriosclerosis, inflammation, apoplexis, angina pectoris, restenosis after angioplasty, claudicatio intermittens, tumours, tumour diseases and/or tumour metastases.

Inventors:
Medellsky, Werner
Uraszik, Horst
Dolsh, Dieter
Tsar Krachidis, Christos
Glitz, Johannes
Burns, christopher
Application Number:
JP2002516259A
Publication Date:
February 19, 2004
Filing Date:
July 03, 2001
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
A61K31/165; A61K31/18; A61K31/27; A61K31/41; A61K31/4245; A61K31/4402; A61K31/445; A61P7/02; A61P9/08; A61P9/10; A61P29/00; A61P35/00; A61P35/04; A61P43/00; C07C257/18; C07C311/16; C07C317/44; C07C327/26; C07C327/28; C07D213/30; C07D257/04; C07D271/06; C07D211/46; (IPC1-7): C07C311/16; A61K31/165; A61K31/18; A61K31/27; A61K31/41; A61K31/4245; A61K31/4402; A61K31/445; A61P7/02; A61P9/08; A61P9/10; A61P29/00; A61P35/00; A61P35/04; A61P43/00; C07C317/44; C07C327/26; C07C327/28; C07D211/46; C07D213/30; C07D257/04; C07D271/06
Attorney, Agent or Firm:
Kiyoji Kuzuwa