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Title:
リポキシゲナーゼ阻害剤
Document Type and Number:
Japanese Patent JP6484201
Kind Code:
B2
Abstract:
The disclosure provides bisindole suitable for inhibiting lipoxygenases or Aβ-formation, and treating associated diseases, such as Alzheimer's disease. The bisindoles are indolo[2,3-b]carbazole derivatives, and may be administered to a patient as part of a pharmaceutical formulation.

Inventors:
John Lynn
Application Number:
JP2016152905A
Publication Date:
March 13, 2019
Filing Date:
August 03, 2016
Export Citation:
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Assignee:
SRI International
International Classes:
A61K31/407; A61K31/439; A61K31/445; A61K31/496; A61K31/5513; A61K31/7072; A61K31/7076; A61K31/708; A61P25/28; A61P43/00; C12N5/00
Domestic Patent References:
JP6034853B2
Foreign References:
WO2006105196A1
US20040043965
WO2010118339A1
WO2006047716A1
WO2006083458A1
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yoshie Sakurada
Yousuke Kawasaki
Takuya Gomibuchi
Toshikazu Imato
Yoichi Iino
Yusuke Ichikawa
Masahiro Moriyama
Yoshikazu Iwase
Yasufumi Shiroyama



 
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