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Title:
MYSTファミリーヒストンアセチルトランスフェラーゼ阻害剤
Document Type and Number:
Japanese Patent JP2021504314
Kind Code:
A
Abstract:
本開示は、化合物、その薬学的に許容される組成物及びそれを使用する方法を提供する。

Inventors:
Harvey, Darren Martin
Campbell, John Emerson
Duncan, Kenneth William
Application Number:
JP2020527906A
Publication Date:
February 15, 2021
Filing Date:
November 29, 2018
Export Citation:
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Assignee:
EPIZIM, INCORPORATED
International Classes:
C07D233/64; A61K31/415; A61K31/4155; A61K31/4164; A61K31/4178; A61K31/4192; A61K31/4196; A61K31/422; A61K31/427; A61K31/4402; A61K31/4439; A61K31/454; A61K31/4545; A61K31/46; A61K31/496; A61K31/5377; A61P35/00; A61P43/00; C07D205/04; C07D207/08; C07D211/24; C07D213/56; C07D223/04; C07D223/06; C07D231/12; C07D233/84; C07D241/04; C07D249/06; C07D265/30; C07D401/12; C07D401/14; C07D403/12; C07D403/14; C07D405/12; C07D405/14; C07D409/12; C07D413/06; C07D413/12; C07D417/12; C07D451/02; C07D493/08
Domestic Patent References:
JP2018524294A2018-08-30
JP2020502064A2020-01-23
JP2022065101A2022-04-26
Other References:
JONATHAN B.BAELL ET AL.: "Inhibitors of histone acetyltransferases KAT6A/B induce senscence and arrest tumour growth", NATURE, vol. 560巻, JPN7022005222, 2018, pages 253 - 257, XP036563466, ISSN: 0004913736, DOI: 10.1038/s41586-018-0387-5
Attorney, Agent or Firm:
Hidesaku Yamamoto
Natsuki Morishita
Takatoshi Iida
Daisuke Ishikawa
Kensaku Yamamoto