Title:
MEDICALLY USEFUL 3*4*55TRIMETHOXYBFNZENE DERIVATIVE
Document Type and Number:
Japanese Patent JPS53135945
Kind Code:
A
Abstract:
Compounds of the formula I (I) wherein m and n are 0, 1 or 2, X represents oxygen, imino, benzylimino, or morpholinoethylimino, Y represents CO, CONH, COO or SO2, and NR1R2 represents a dimethylamino, diethylamino, dipropylamino, dibutylamino, allylamino, isobutenylamino, cyclopentylamino, cyclohexylamino, cycloheptylamino, cyclooctylamino, N-methyl N-cyclopentylamino, N-methyl N-cyclohexylamino, N-allyl N-cyclohexylamino, adamantylamino, diethoxyethylamino, dimethylaminoethylamino, dimethylaminopropylamino, N-methyl N-dimethylaminopropyl-amino, benzylamino, 3,4,5-trimethoxybenzylamino, phenethylamino, p-chlorophenethylamino, tetrahydrofurfurylamino, tetrahydropyranylmethylamino, pyrrolidino, isoxazolidinyl, piperidino, 4-hydroxypiperidino, 4-m-chlorophenyl-4-hydroxypiperidino, homopiperidino, 1,2,3,6-tetrahydropyridyl, morpholino, 2-methylmorpholino, 2,6-dimethylmorpholino, 2-morpholinoethylamino, thiamorpholino, piperazino, 4-methylpiperazino, 4-( alpha -m-chlorophenyl-benzyl)-piperazino, 4-(3,4,5-trimethoxyphenylaminocarbonyl)-piperazino, 4-(3,4,5-trimethoxyphenylaminocarbonylmethyl)-piperazino, 4-phenylpiperazino, 4-m-trifluoromethylphenyl-piperazino, 4-piperidinocarbonylmethyl-piperazino, 1,2,3,4-tetrahydroquinolyl, 1,2,3,4-tetrahydroisoquinolyl, (7-chloro-4-quinolyl)-amino, 1,2,3,4-tetrahydrobenzoxazinyl or 1,2,3,4-tetrahydro-6-chlorobenzoxazinyl group, and their pharmaceutically acceptable acid addition salts are novel and are therapeutically useful, in particular as tranquillizers, myorelaxants and anticonvulsants.
Inventors:
MOORISU JIYURIE
GABURIERU MEIYAARU
RIYUSHIAN RAKA
KURISUCHIYAN JIYAN MARII WAROR
GABURIERU MEIYAARU
RIYUSHIAN RAKA
KURISUCHIYAN JIYAN MARII WAROR
Application Number:
JP209578A
Publication Date:
November 28, 1978
Filing Date:
January 13, 1978
Export Citation:
Assignee:
METABIO JOULLIE SA
International Classes:
A61K31/135; A61K31/165; A61K31/215; A61K31/22; A61K31/255; A61K31/27; A61K31/435; A61K31/535; A61K31/536; A61K31/5375; A61K31/538; A61P25/00; A61P25/08; A61P25/24; A61P25/26; A61K31/16; C07C67/00; C07C219/06; C07C225/06; C07C227/00; C07C227/02; C07C229/18; C07C231/00; C07C231/02; C07C231/10; C07C235/20; C07C239/00; C07C273/10; C07C275/34; C07C301/00; C07C303/34; C07C303/38; C07C307/10; C07D211/46; C07D211/52; C07D211/70; C07D215/06; C07D215/08; C07D215/42; C07D215/44; C07D217/02; C07D217/06; C07D261/02; C07D265/30; C07D265/36; C07D295/088; C07D295/13; C07D295/15; C07D295/185; C07D295/205; C07D295/215; C07D295/24; C07D295/26; C07D295/28; C07D307/14; C07D309/04; C07D309/14; (IPC1-7): A61K31/16; A61K31/215; A61K31/255; A61K31/27; A61K31/435; A61K31/535; C07C93/187; C07C97/02; C07C101/16; C07C103/44; C07C127/19; C07C147/14; C07D295/08; C07D295/12; C07D295/16