Title:
非ヌクレオシドHIV-1逆転写酵素インヒビターの製造方法及び中間体
Document Type and Number:
Japanese Patent JP2005538971
Kind Code:
A
Abstract:
A process and novel intermediates for making compounds of the formula I: wherein: R<2 >is selected from the group consisting of H, F, Cl, C1-4 alkyl, C3-4 cycloalkyl and CF3; R<4 >is H or Me; R<5 >is H, Me or Et, with the proviso that R<4 >and R<5 >are not both Me, and if R<4 >is Me then R<5 >cannot be Et; R<11 >is Me, Et, cyclopropyl, propyl, isopropyl, or cyclobutyl; and Q is selected from the group consisting of:
Inventors:
Bussakka Karl A
Ericsson Magnus Sea
Kim Ji Yang
Ericsson Magnus Sea
Kim Ji Yang
Application Number:
JP2004517701A
Publication Date:
December 22, 2005
Filing Date:
June 20, 2003
Export Citation:
Assignee:
Boehringer Ingelheim Pharmaceuticals, Inc.
International Classes:
C07B61/00; C07D471/14; C07F9/6524; C07D471/04; (IPC1-7): C07D471/04; C07F9/6524
Attorney, Agent or Firm:
Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama