Title:
ピリミジニルシクロペンタン化合物の調製方法
Document Type and Number:
Japanese Patent JP6857219
Kind Code:
B2
Abstract:
The present invention relates to a process for the preparation of a compound of formula (I)wherein R1 is as defined herein, which is useful as an intermediate in the preparation of active pharmaceutical compounds.
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Inventors:
Han Siding
Reinhard Lanez
Michelangelo Scalone
Francis gosselin
Reinhard Lanez
Michelangelo Scalone
Francis gosselin
Application Number:
JP2019155667A
Publication Date:
April 14, 2021
Filing Date:
August 28, 2019
Export Citation:
Assignee:
Ef Hoffman-La Roche Akchengezel Shaft
Genentech, Incorporated
Genentech, Incorporated
International Classes:
C07C271/22; A61K31/517; A61P35/00; C07C269/06
Domestic Patent References:
| JP2009542723A | ||||
| JP2015520165A |
Other References:
Blake, James F.; Xu, Rui; Bencsik, Josef R.; Xiao, Dengming; Kallan, Nicholas C.; Schlachter, Stephe,Discovery and Preclinical Pharmacology of a Selective ATP-Competitive Akt Inhibitor (GDC-0068) for the Treatment of Human Tumors,Journal of Medicinal Chemistry,2012年,55(18),8110-8127
Elaridi, Jomana; Thaqi, Ali; Prosser, Andrew; Jackson, W. Roy; Robinson, Andrea J.,An enantioselective synthesis of β2-amino acid derivatives,Tetrahedron: Asymmetry,2005年,16(7),1309-1319
Elaridi, Jomana; Thaqi, Ali; Prosser, Andrew; Jackson, W. Roy; Robinson, Andrea J.,An enantioselective synthesis of β2-amino acid derivatives,Tetrahedron: Asymmetry,2005年,16(7),1309-1319
Attorney, Agent or Firm:
Hidesaku Yamamoto
Natsuki Morishita
Natsuki Morishita