Title:
置換オクタノイルアミドの調製方法
Document Type and Number:
Japanese Patent JP4900755
Kind Code:
B2
Abstract:
Compounds of formula (II) are simultaneously halogenated in the 5 position and hydroxylated in the 4 position under lactonization, the halolactone is converted into a hydroxylactone and then the hydroxy group into a leaving group, the leaving group is replaced with azide, the lactone amidated and then the azide converted to the amine group, in order to obtain compounds of formula (I).
Inventors:
Herolt, peter
Stutz, Stephan
Felix, Spintorer
Stutz, Stephan
Felix, Spintorer
Application Number:
JP2002507765A
Publication Date:
March 21, 2012
Filing Date:
June 26, 2001
Export Citation:
Assignee:
Novartis Pharma AG
International Classes:
C07C231/12; C07B61/00; C07C57/42; C07C59/64; C07C59/68; C07C69/734; C07C231/02; C07C231/18; C07C237/20; C07C247/12; C07D207/33; C07D303/38; C07D303/40; C07D307/33; C07B53/00; C07D207/32
Domestic Patent References:
| JP8081430A | ||||
| JP8053434A |
Attorney, Agent or Firm:
Hajime Tsukuni
Fusayuki Saito
Satoko Ito
Keiko Ozawa
Fumio Shinoda
Koshiro Tsukuda
Fusayuki Saito
Satoko Ito
Keiko Ozawa
Fumio Shinoda
Koshiro Tsukuda