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Title:
MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONIST
Document Type and Number:
Japanese Patent JP2011162556
Kind Code:
A
Abstract:

To provide muscarinic acetylcholine receptor antagonists and methods of using them.

There are provided: (Endo)-3-(2-cyano-2,2-diphenyl-ethyl)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane bromide; (Endo)-3-(2-cyano-2,2-diphenyl-ethyl)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane iodide; and methods of using them.


Inventors:
BUSCH-PETERSEN JAKOB
PALOVICH MICHAEL R
WAN ZEHONG
YAN HONGXING
ZHU CHONGJIE
Application Number:
JP2011109756A
Publication Date:
August 25, 2011
Filing Date:
May 16, 2011
Export Citation:
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Assignee:
GLAXO GROUP LTD
International Classes:
C07D451/02; A61K9/12; A61K31/437; A61K31/46; A61P1/04; A61P11/00; A61P11/06; A61P13/10; A61P37/08; A61P43/00
Domestic Patent References:
JPH06505718A1994-06-30
JPH0920758A1997-01-21
JPH05501554A1993-03-25
JP4796552B22011-10-19
Foreign References:
US2800478A1957-07-23
US2800481A1957-07-23
WO2003033495A12003-04-24
WO1995015951A11995-06-15
Attorney, Agent or Firm:
Aoyama Aoi
Takuji Yamada
Michiko Matsutani
Yasushi Ochiai