Title:
新規フェニルアラニン誘導体
Document Type and Number:
Japanese Patent JP4784803
Kind Code:
B2
Abstract:
Phenylalanine derivatives of the following formula and analogues thereof have an antagonistic activity to alpha 4 beta 7 integrin and a selectivity toward alpha 4 beta 1 integrin. They are used as therapeutic agents for various diseases to which alpha 4 beta 7 integrin relates.
Inventors:
Yasuhiro Tanaka
Toshihiko Yoshimura
Tomoko Ejima
Mitsuhiko Kojima
Eiji Nakanishi
Hiroyuki Izawa
Yuko Satake
Suzuki Shiniku
Suzuki Manabu
Murata Masahiro
Toshihiko Yoshimura
Tomoko Ejima
Mitsuhiko Kojima
Eiji Nakanishi
Hiroyuki Izawa
Yuko Satake
Suzuki Shiniku
Suzuki Manabu
Murata Masahiro
Application Number:
JP2001549342A
Publication Date:
October 05, 2011
Filing Date:
December 26, 2000
Export Citation:
Assignee:
AJINOMOTO CO.,LTD.
International Classes:
C07C233/63; A61K31/198; A61K31/397; A61K31/433; A61K31/445; A61K31/472; A61K31/495; A61K31/505; A61K31/5375; A61K31/54; A61K31/55; A61P1/04; A61P3/10; A61P35/00; A61P35/04; A61P43/00; C07C243/36; C07C243/38; C07C255/65; C07C281/06; C07C311/21; C07C311/39; C07C311/44; C07C311/46; C07C321/28; C07C323/40; C07D205/04; C07D207/12; C07D207/14; C07D211/32; C07D211/46; C07D211/58; C07D211/62; C07D217/06; C07D223/04; C07D233/52; C07D239/38; C07D285/06; C07D295/18; C07D295/185; C07D295/22; C07D295/32
Domestic Patent References:
JP2003524614A | 2003-08-19 |
Attorney, Agent or Firm:
Minoru Nakamura
Fumiaki Otsuka
Sadao Kumakura
Shishido Kaichi
Hideto Takeuchi
Toshio Imajo
Nobuo Ogawa
Village shrine Atsuo
Takaki Nishijima
Atsushi Hakoda
Fumiaki Otsuka
Sadao Kumakura
Shishido Kaichi
Hideto Takeuchi
Toshio Imajo
Nobuo Ogawa
Village shrine Atsuo
Takaki Nishijima
Atsushi Hakoda