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Title:
新規フェニルアラニン誘導体
Document Type and Number:
Japanese Patent JP4784803
Kind Code:
B2
Abstract:
Phenylalanine derivatives of the following formula and analogues thereof have an antagonistic activity to alpha 4 beta 7 integrin and a selectivity toward alpha 4 beta 1 integrin. They are used as therapeutic agents for various diseases to which alpha 4 beta 7 integrin relates.

Inventors:
Yasuhiro Tanaka
Toshihiko Yoshimura
Tomoko Ejima
Mitsuhiko Kojima
Eiji Nakanishi
Hiroyuki Izawa
Yuko Satake
Suzuki Shiniku
Suzuki Manabu
Murata Masahiro
Application Number:
JP2001549342A
Publication Date:
October 05, 2011
Filing Date:
December 26, 2000
Export Citation:
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Assignee:
AJINOMOTO CO.,LTD.
International Classes:
C07C233/63; A61K31/198; A61K31/397; A61K31/433; A61K31/445; A61K31/472; A61K31/495; A61K31/505; A61K31/5375; A61K31/54; A61K31/55; A61P1/04; A61P3/10; A61P35/00; A61P35/04; A61P43/00; C07C243/36; C07C243/38; C07C255/65; C07C281/06; C07C311/21; C07C311/39; C07C311/44; C07C311/46; C07C321/28; C07C323/40; C07D205/04; C07D207/12; C07D207/14; C07D211/32; C07D211/46; C07D211/58; C07D211/62; C07D217/06; C07D223/04; C07D233/52; C07D239/38; C07D285/06; C07D295/18; C07D295/185; C07D295/22; C07D295/32
Domestic Patent References:
JP2003524614A2003-08-19
Attorney, Agent or Firm:
Minoru Nakamura
Fumiaki Otsuka
Sadao Kumakura
Shishido Kaichi
Hideto Takeuchi
Toshio Imajo
Nobuo Ogawa
Village shrine Atsuo
Takaki Nishijima
Atsushi Hakoda