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Title:
NOVEL PYRAZOLO-BENZODIAZEPINE DERIVATIVE AND PREPARATION THEREOF
Document Type and Number:
Japanese Patent JPS58103389
Kind Code:
A
Abstract:

NEW MATERIAL:A 4-amino pyrazolo[3,4-b][1,5]benzodiazepine derivative (acid addition salt) of formulaI(R is H, methyl of phenyl; X is H or chlorine).

USE: A psychotropic agent.

PROCESS: (A) A 4-amino-3-cyano-[1H]-1,5-benzodiazepine of formula II or a chlorine derivative or a hydrochloride thereof is usually reacted with (B) preferably 2W10mol, based on one mole component (A), hydrazine of the formula NH2NH-R or an N-substituted hydrazine in a solvent, e.g. water or methanol, for several hours under heating.


Inventors:
TAKAGI KANAME
OKAMOTO YOSHIHISA
Application Number:
JP20136681A
Publication Date:
June 20, 1983
Filing Date:
December 12, 1981
Export Citation:
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Assignee:
ZERIA PHARM CO LTD
International Classes:
C07D487/04; A61K31/55; A61P25/00; (IPC1-7): A61K31/55; C07D487/04
Attorney, Agent or Firm:
Tsunemitsu Yamada



 
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